The synthetic purine reversine selectively induces cell death of cancer cells

J Cell Biochem. 2012 Oct;113(10):3207-17. doi: 10.1002/jcb.24197.

Abstract

The synthetic purine reversine has been shown to possess a dual activity as it promotes the de-differentiation of adult cells, including fibroblasts, into stem-cell-like progenitors, but it also induces cell growth arrest and ultimately cell death of cancer cells, suggesting its possible application as an anti-cancer agent. Aim of this study was to investigate the mechanism underneath reversine selectivity in inducing cell death of cancer cells by a comparative analysis of its effects on several tumor cells and normal dermal fibroblasts. We found that reversine is lethal for all cancer cells studied as it induces cell endoreplication, a process that malignant cells cannot effectively oppose due to aberrations in cell cycle checkpoints. On the other hand, normal cells, like dermal fibroblasts, can control reversine activity by blocking the cell cycle, entering a reversible quiescent state. However, they can be induced to become sensitive to the molecule when key cell cycle proteins, e.g., p53, are silenced.

MeSH terms

  • Antineoplastic Agents / pharmacology*
  • Benzothiazoles / pharmacology
  • Blotting, Western
  • Caspases / metabolism
  • Cell Cycle Checkpoints
  • Cell Death
  • Cell Dedifferentiation
  • Cell Proliferation
  • Cell Shape / drug effects
  • Cell Survival
  • Endoreduplication
  • Enzyme Activation
  • Fibroblasts / drug effects
  • Fibrosarcoma / genetics
  • Fibrosarcoma / metabolism
  • Fibrosarcoma / pathology
  • Flow Cytometry
  • Gene Silencing
  • HeLa Cells
  • Humans
  • Morpholines / pharmacology*
  • Purines / pharmacology*
  • RNA, Small Interfering / genetics
  • RNA, Small Interfering / metabolism
  • Toluene / analogs & derivatives
  • Toluene / pharmacology
  • Tumor Suppressor Protein p53 / antagonists & inhibitors
  • Tumor Suppressor Protein p53 / genetics
  • Tumor Suppressor Protein p53 / metabolism*

Substances

  • Antineoplastic Agents
  • Benzothiazoles
  • Morpholines
  • Purines
  • RNA, Small Interfering
  • Tumor Suppressor Protein p53
  • Toluene
  • pifithrin
  • Caspases
  • 2-(4-morpholinoanilino)-6-cyclohexylaminopurine