Effects of exogenous cholecystokinin octapeptide on acquisition of naloxone precipitated withdrawal induced conditioned place aversion in rats

PLoS One. 2012;7(7):e41860. doi: 10.1371/journal.pone.0041860. Epub 2012 Jul 27.

Abstract

Cholecystokinin octapeptide (CCK-8), a gut-brain peptide, regulates a variety of physiological behavioral processes. Previously, we reported that exogenous CCK-8 attenuated morphine-induced conditioned place preference, but the possible effects of CCK-8 on aversively motivated drug seeking remained unclear. To investigate the effects of endogenous and exogenous CCK on negative components of morphine withdrawal, we evaluated the effects of CCK receptor antagonists and CCK-8 on the naloxone-precipitated withdrawal-induced conditioned place aversion (CPA). The results showed that CCK2 receptor antagonist (LY-288,513, 10 µg, i.c.v.), but not CCK1 receptor antagonist (L-364,718, 10 µg, i.c.v.), inhibited the acquisition of CPA when given prior to naloxone (0.3 mg/kg) administration in morphine-dependent rats. Similarly, CCK-8 (0.1-1 µg, i.c.v.) significantly attenuated naloxone-precipitated withdrawal-induced CPA, and this inhibitory function was blocked by co-injection with L-364,718. Microinjection of L-364,718, LY-288,513 or CCK-8 to saline pretreated rats produced neither a conditioned preference nor aversion, and the induction of CPA by CCK-8 itself after morphine pretreatments was not significant. Our study identifies a different role of CCK1 and CCK2 receptors in negative affective components of morphine abstinence and an inhibitory effect of exogenous CCK-8 on naloxone-precipitated withdrawal-induced CPA via CCK1 receptor.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Conditioning, Psychological / drug effects*
  • Devazepide / pharmacology
  • Male
  • Morphine Dependence / drug therapy
  • Morphine Dependence / etiology
  • Morphine Dependence / metabolism
  • Morphine Dependence / psychology
  • Naloxone / pharmacology*
  • Pyrazoles / pharmacology
  • Rats
  • Rats, Wistar
  • Receptors, Cholecystokinin / antagonists & inhibitors
  • Sincalide / metabolism
  • Sincalide / pharmacology*
  • Sincalide / therapeutic use
  • Spatial Behavior / drug effects*
  • Substance Withdrawal Syndrome / drug therapy*
  • Substance Withdrawal Syndrome / etiology
  • Substance Withdrawal Syndrome / metabolism
  • Substance Withdrawal Syndrome / psychology*

Substances

  • Pyrazoles
  • Receptors, Cholecystokinin
  • 1-(4-bromophenylaminocarbonyl)-4,5-diphenyl-3-pyrazolidinone
  • Naloxone
  • Devazepide
  • Sincalide

Grants and funding

This study was supported in part by grants from the Natural Science Foundation of China (www.nsfc.gov.cn) (No. 81172900, 30672355), the Applied Basic Research Key Program of Hebei Province (No. 10966911D) and the Natural Science Foundation of Hebei Province (www.hensf.gov.cn) (No. C2007000826). The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript.