Characterization of novel genomic alterations and therapeutic approaches using acute megakaryoblastic leukemia xenograft models

J Exp Med. 2012 Oct 22;209(11):2017-31. doi: 10.1084/jem.20121343. Epub 2012 Oct 8.

Abstract

Acute megakaryoblastic leukemia (AMKL) is a heterogeneous disease generally associated with poor prognosis. Gene expression profiles indicate the existence of distinct molecular subgroups, and several genetic alterations have been characterized in the past years, including the t(1;22)(p13;q13) and the trisomy 21 associated with GATA1 mutations. However, the majority of patients do not present with known mutations, and the limited access to primary patient leukemic cells impedes the efficient development of novel therapeutic strategies. In this study, using a xenotransplantation approach, we have modeled human pediatric AMKL in immunodeficient mice. Analysis of high-throughput RNA sequencing identified recurrent fusion genes defining new molecular subgroups. One subgroup of patients presented with MLL or NUP98 fusion genes leading to up-regulation of the HOX A cluster genes. A novel CBFA2T3-GLIS2 fusion gene resulting from a cryptic inversion of chromosome 16 was identified in another subgroup of 31% of non-Down syndrome AMKL and strongly associated with a gene expression signature of Hedgehog pathway activation. These molecular data provide useful markers for the diagnosis and follow up of patients. Finally, we show that AMKL xenograft models constitute a relevant in vivo preclinical screening platform to validate the efficacy of novel therapies such as Aurora A kinase inhibitors.

MeSH terms

  • 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine / analogs & derivatives
  • 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine / pharmacology
  • Aged
  • Amino Acid Sequence
  • Animals
  • Aurora Kinase A
  • Aurora Kinases
  • Azepines / pharmacology
  • Base Sequence
  • Female
  • Gene Expression Profiling
  • Genomics / methods*
  • High-Throughput Nucleotide Sequencing / methods
  • Humans
  • Infant
  • Kaplan-Meier Estimate
  • Kruppel-Like Transcription Factors / genetics
  • Leukemia, Megakaryoblastic, Acute / drug therapy*
  • Leukemia, Megakaryoblastic, Acute / genetics*
  • Leukemia, Megakaryoblastic, Acute / pathology
  • Male
  • Mice
  • Mice, SCID
  • Middle Aged
  • Molecular Sequence Data
  • Oligonucleotide Array Sequence Analysis
  • Oncogene Proteins, Fusion / genetics
  • Protein Serine-Threonine Kinases / antagonists & inhibitors
  • Pyrimidines / pharmacology
  • Repressor Proteins / genetics
  • Xenograft Model Antitumor Assays*

Substances

  • 2-methyl-1-((4-methyl-5-isoquinolinyl)sulfonyl)homopiperazine
  • Azepines
  • CBFA2T2 myeloid-transforming gene-related protein
  • CBFA2T3-GLIS2 fusion protein, human
  • GLIS2 protein, human
  • Kruppel-Like Transcription Factors
  • MLN 8237
  • Oncogene Proteins, Fusion
  • Pyrimidines
  • Repressor Proteins
  • 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine
  • Aurka protein, mouse
  • Aurora Kinase A
  • Aurora Kinases
  • Protein Serine-Threonine Kinases