Phorbol 12-myristate 13-acetate (PMA) increases the expression of the nerve growth factor (NGF) gene in mouse L-929 fibroblasts

FEBS Lett. 1990 Mar 12;262(1):42-4. doi: 10.1016/0014-5793(90)80149-d.

Abstract

The rise of the NGF mRNA pool which takes place following exposure of L-929 fibroblasts to serum was prevented in the presence of 5 microM K-252a, a compound which inhibits several species of protein kinase activities. To characterize further this phenomenon, L-929 cells growing in a serum-free medium were exposed to cyclic nucleotide analogs, to a divalent cation ionophore or to the phorbol ester PMA. Only this latter compound induced an enhancement of the NGF mRNA pool, suggesting an involvement of protein kinase C in the upregulation of the NGF transcripts. The effects of PMA or serum also require a synthesis of protein since the level of NGF transcripts remained stable in the presence of cycloheximide.

MeSH terms

  • Animals
  • Blood Physiological Phenomena
  • Carbazoles / pharmacology
  • Fibroblasts / metabolism
  • Gene Expression / drug effects*
  • Indole Alkaloids
  • Mice
  • Nerve Growth Factors / genetics*
  • Protein Biosynthesis
  • Protein Kinase C / physiology
  • RNA, Messenger / analysis
  • Tetradecanoylphorbol Acetate / pharmacology*

Substances

  • Carbazoles
  • Indole Alkaloids
  • Nerve Growth Factors
  • RNA, Messenger
  • staurosporine aglycone
  • Protein Kinase C
  • Tetradecanoylphorbol Acetate