RS-WebPredictor: a server for predicting CYP-mediated sites of metabolism on drug-like molecules

Bioinformatics. 2013 Feb 15;29(4):497-8. doi: 10.1093/bioinformatics/bts705. Epub 2012 Dec 14.

Abstract

Summary: Regioselectivity-WebPredictor (RS-WebPredictor) is a server that predicts isozyme-specific cytochrome P450 (CYP)-mediated sites of metabolism (SOMs) on drug-like molecules. Predictions may be made for the promiscuous 2C9, 2D6 and 3A4 CYP isozymes, as well as CYPs 1A2, 2A6, 2B6, 2C8, 2C19 and 2E1. RS-WebPredictor is the first freely accessible server that predicts the regioselectivity of the last six isozymes. Server execution time is fast, taking on average 2s to encode a submitted molecule and 1s to apply a given model, allowing for high-throughput use in lead optimization projects.

Availability: RS-WebPredictor is accessible for free use at http://reccr.chem.rpi.edu/Software/RS-WebPredictor/

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Algorithms
  • Cinnarizine / chemistry
  • Cinnarizine / metabolism
  • Cytochrome P-450 Enzyme System / metabolism*
  • Isoenzymes / metabolism
  • Software*

Substances

  • Isoenzymes
  • Cinnarizine
  • Cytochrome P-450 Enzyme System