The Akt DUBbed InAktive

Sci Signal. 2013 Jan 8;6(257):pe1. doi: 10.1126/scisignal.2003864.

Abstract

Akt is a central node in the phosphoinositide-3 kinase-Akt-mammalian target of rapamycin pathway and is activated by a multistep process in response to growth factor stimulation. An additional layer of posttranslational modification has emerged as a new paradigm in the regulation of Akt. The identification of an E3 ligase for Lys(63)-linked ubiquitination of Akt has now been complemented with the discovery of the tumor suppressor cylindromatosis as a deubiquitinating enzyme (DUB) for Akt. Thus, like phosphorylation and dephosphorylation, cycles of ubiquitination and deubiquitination provide additional on-off switches that keep Akt activity in balance, and disturbances in this balance have pathological consequences.

MeSH terms

  • Deubiquitinating Enzyme CYLD
  • Gene Expression Regulation, Neoplastic / physiology*
  • Humans
  • Intercellular Signaling Peptides and Proteins / metabolism
  • Models, Biological*
  • Proto-Oncogene Proteins c-akt / genetics
  • Proto-Oncogene Proteins c-akt / metabolism*
  • Signal Transduction / physiology*
  • Tumor Suppressor Proteins / metabolism*
  • Ubiquitination / physiology*

Substances

  • Intercellular Signaling Peptides and Proteins
  • Tumor Suppressor Proteins
  • Proto-Oncogene Proteins c-akt
  • CYLD protein, human
  • Deubiquitinating Enzyme CYLD