PLA/PEG-PPG-PEG/dexamethasone implant prepared by hot-melt extrusion for controlled release of immunosuppressive drug to implantable medical devices, Part 2: in vivo evaluation

Drug Deliv. 2013 Apr-May;20(3-4):134-42. doi: 10.3109/10717544.2013.801049.

Abstract

Hot-melt extrusion (HME) plays an important role in preparing implants as local drug delivery systems in pharmaceutical fields. Here, a new PLA/PEG-PPG-PEG/Dexamethasone (PLA/F68/Dex) implant prepared by HME has been developed. Importantly, the implant was successfully achieved to control release of immunosuppressive drug to an implanted device. In particular, this implant has not been reported previously in pharmaceutical fields. FTIR and XRD were adopted to investigate the properties of the samples. The in vivo release study showed that the maximum value of Dex release from the implants was approximately 50% at 1 month. The in vivo degradation behavior was determined by UV spectrophotometer and scanning electron microscopy studies, and the weight loss rate of the implants were up to 25% at 1 month. Furthermore, complete blood count (CBC) test, serum chemistry and major organs were performed, and there is no significant lesion and side effects observed in these results. Therefore, the results elucidated that the new PLA/F68/Dex implant prepared by HME could deliver an immunosuppressive drug to control the inflammatory reaction at the implant site.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Delayed-Action Preparations / administration & dosage
  • Delayed-Action Preparations / chemical synthesis
  • Dexamethasone / administration & dosage
  • Dexamethasone / chemical synthesis*
  • Drug Evaluation, Preclinical / methods
  • Hot Temperature*
  • Immunosuppressive Agents / administration & dosage
  • Immunosuppressive Agents / chemical synthesis*
  • Infusion Pumps, Implantable*
  • Male
  • Polyethylene Glycols / administration & dosage
  • Polyethylene Glycols / chemical synthesis*
  • Propylene Glycols / administration & dosage
  • Propylene Glycols / chemical synthesis*
  • Rats
  • Rats, Sprague-Dawley
  • X-Ray Diffraction

Substances

  • Delayed-Action Preparations
  • Immunosuppressive Agents
  • Propylene Glycols
  • poly(ethylene glycol)-block-poly(propylene glycol)-block-poly(ethylene glycol) copolymer
  • Polyethylene Glycols
  • Dexamethasone