Enhancement of skin radical scavenging activity and stratum corneum lipids after the application of a hyperforin-rich cream

Eur J Pharm Biopharm. 2014 Feb;86(2):227-33. doi: 10.1016/j.ejpb.2013.06.016. Epub 2013 Jun 26.

Abstract

Hyperforin is well-known for its anti-inflammatory, anti-tumor, anti-bacterial, and antioxidant properties. The application of a hyperforin-rich verum cream could strengthen the skin barrier function by reducing radical formation and stabilizing stratum corneum lipids. Here, it was investigated whether topical treatment with a hyperforin-rich cream increases the radical protection of the skin during VIS/NIR irradiation. Skin lipid profile was investigated applying HPTLC on skin lipid extracts. Furthermore, the absorption- and scattering coefficients, which influence radical formation, were determined. 11 volunteers were included in this study. After a single cream application, VIS/NIR-induced radical formation could be completely inhibited by both verum and placebo showing an immediate protection. After an application period of 4weeks, radical formation could be significantly reduced by 45% following placebo application and 78% after verum application showing a long-term protection. Furthermore, the skin lipids in both verum and placebo groups increased directly after a single cream application but only significantly for ceramide [AP], [NP1], and squalene. After long-term cream application, concentration of cholesterol and the ceramides increased, but no significance was observed. These results indicate that regular application of the hyperforin-rich cream can reduce radical formation and can stabilize skin lipids, which are responsible for the barrier function.

Keywords: Electron paramagnetic resonance spectroscopy; High performance thin layer chromatography; Hypericum perforatum; Skin lipid profile; St. John’s Wort.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Anti-Inflammatory Agents / administration & dosage*
  • Anti-Inflammatory Agents / metabolism
  • Ceramides / metabolism
  • Female
  • Free Radical Scavengers / administration & dosage*
  • Free Radical Scavengers / metabolism
  • Humans
  • Lipids
  • Male
  • Phloroglucinol / administration & dosage
  • Phloroglucinol / analogs & derivatives*
  • Phloroglucinol / metabolism
  • Skin / drug effects*
  • Skin / metabolism
  • Skin Absorption
  • Skin Cream / metabolism
  • Skin Cream / therapeutic use*
  • Terpenes / administration & dosage*
  • Terpenes / metabolism
  • Young Adult

Substances

  • Anti-Inflammatory Agents
  • Ceramides
  • Free Radical Scavengers
  • Lipids
  • Terpenes
  • Phloroglucinol
  • hyperforin