Overcoming cancer cell resistance to VSV oncolysis with JAK1/2 inhibitors

Cancer Gene Ther. 2013 Oct;20(10):582-9. doi: 10.1038/cgt.2013.55. Epub 2013 Sep 13.

Abstract

Oncolytic vesicular stomatitis virus (VSV) has potent antitumor activity but some cancer cells are resistant to VSV killing, either constitutively or due to type I interferon (IFN) inducing an antiviral state in the cells. Here, we evaluated VSV oncolysis of a panel of human head and neck cancer cells and showed that VSV resistance in SCC25 and SCC15 cells could be reversed with Janus kinase (JAK) 1/2 inhibitors (JAK inhibitor I and ruxolitinib). Pre-treatment of cells with JAK1/2 inhibitors before or in conjunction with VSV enhanced viral infection, spread and progeny yield (100- to 1000-fold increase). In contrast, inhibitors of histone deacetylase (LBH589), phosphatidylinositol 3-kinase (GDC-0941, LY294002), mammalian target of rapamycin (rapamycin) or signal transducer and activator of transcription 3 (STAT3 inhibitor VII) were ineffective. Compared with VSV-sensitive SW579 cells, IFNα/β responsive antiviral genes (IRF-9, IRF-7, OAS1 but not MxA) are constitutively expressed in SCC25 cells. Pretreatment with JAK inhibitors reduced mRNA levels of these genes, increasing VSV expression in the cells. Interestingly, 1 h of drug exposure was sufficient to reverse SCC25 resistance to VSV and was still effective if virus was added 24 h later. Overall, we show here that JAK inhibitor I and ruxolitinib (Jakafi) can reverse resistance to VSV, supporting the rationale to incorporate JAK1/2 inhibitors in future VSV virotherapy trials.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Carcinoma, Squamous Cell / enzymology
  • Carcinoma, Squamous Cell / immunology
  • Carcinoma, Squamous Cell / therapy*
  • Carcinoma, Squamous Cell / virology*
  • Cell Line, Tumor
  • Head and Neck Neoplasms / enzymology
  • Head and Neck Neoplasms / immunology
  • Head and Neck Neoplasms / therapy*
  • Head and Neck Neoplasms / virology*
  • Humans
  • Interferon-alpha / genetics
  • Interferon-alpha / immunology
  • Interferon-beta / genetics
  • Interferon-beta / immunology
  • Janus Kinase 1 / antagonists & inhibitors*
  • Janus Kinase 1 / biosynthesis
  • Janus Kinase 1 / genetics
  • Janus Kinase 2 / antagonists & inhibitors*
  • Janus Kinase 2 / biosynthesis
  • Janus Kinase 2 / genetics
  • Nitriles
  • Oncolytic Virotherapy / methods*
  • Protein Kinase Inhibitors / pharmacology*
  • Pyrazoles / pharmacology
  • Pyrimidines
  • RNA, Messenger / biosynthesis
  • RNA, Messenger / genetics
  • Signal Transduction
  • Squamous Cell Carcinoma of Head and Neck
  • Vesicular stomatitis Indiana virus / genetics
  • Vesicular stomatitis Indiana virus / metabolism
  • Vesicular stomatitis Indiana virus / physiology*
  • Virus Replication

Substances

  • Interferon-alpha
  • Nitriles
  • Protein Kinase Inhibitors
  • Pyrazoles
  • Pyrimidines
  • RNA, Messenger
  • Interferon-beta
  • ruxolitinib
  • Janus Kinase 1
  • Janus Kinase 2