Biophysical studies of engineered mutant proteins based on calbindin D9k modified in the pseudo EF-hand

Eur J Biochem. 1990 Jan 26;187(2):455-60. doi: 10.1111/j.1432-1033.1990.tb15325.x.

Abstract

The genes for four mutant proteins from calbindin D9k, all with mutations in the N-terminal Ca2+-binding domain (pseudo EF-hand) have been synthesized and expressed in Escherichia coli. The purification scheme has been modified to minimize the formation of deamidated proteins. The set of modifications in the pseudo EF-hand is an attempt to turn this site into a structure resembling an archetypal EF-hand, with its characteristic 113Cd-NMR shift (-80 to -110 ppm) and high calcium-binding constants, whereas the C-terminal Ca2(+)-binding site (EF-hand) is kept intact in all mutant proteins. The mutant proteins studied here all have pseudo EF-hands with a lower calcium-binding constant and a higher calcium off-rate to the pseudo EF-hand than the wild-type protein. From the results obtained it is obvious that proline 20 in the pseudo EF-hand, which has been deleted or replaced by glycine in three of the mutants, has a stabilizing effect on calcium binding to that site. Furthermore, the modifications in the pseudo EF-hand seem to have only a local effect, leaving the tertiary structure of the protein and the calcium-binding properties of the unmodified site virtually unchanged.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alanine
  • Animals
  • Binding Sites
  • Calbindins
  • Calcium / pharmacology
  • Escherichia coli / genetics
  • Escherichia coli / metabolism
  • Gene Expression
  • Glycine
  • Kinetics
  • Magnetic Resonance Spectroscopy / methods
  • Models, Molecular
  • Mutation
  • Proline
  • Protein Conformation
  • Protein Engineering
  • Recombinant Proteins / biosynthesis
  • Recombinant Proteins / isolation & purification
  • S100 Calcium Binding Protein G / biosynthesis
  • S100 Calcium Binding Protein G / genetics*
  • S100 Calcium Binding Protein G / isolation & purification
  • Temperature

Substances

  • Calbindins
  • Recombinant Proteins
  • S100 Calcium Binding Protein G
  • Proline
  • Alanine
  • Calcium
  • Glycine