Tristetraprolin down-regulates IL-23 expression in colon cancer cells

Mol Cells. 2013 Dec;36(6):571-6. doi: 10.1007/s10059-013-0268-6. Epub 2013 Nov 29.

Abstract

Interleukin 23 (IL-23) is an inflammatory cytokine that plays an important role in tumor promotion. Expression of IL-23 is increased in cancer cells and correlates with tumor progression. However, the mechanisms regulating IL-23 expression in cancer cells are still unclear. Here we report that tristetraprolin (TTP), an AU-rich element (ARE)-binding protein, inhibits IL-23 production in CT26 mouse colon cancer cells. Overexpression of TTP decreased the stability of IL-23 mRNA and the expression level of IL-23 in CT26 cells. Conversely, inhibition of TTP by siRNA increased IL-23 production. TTP destabilized a luciferase mRNA reporter containing the IL-23 mRNA 3'UTR, which contains five AREs. Analyses of deletion and point mutants of the IL-23 mRNA 3'UTR demonstrated that the ARE cluster between the third and fifth AREs was responsible for TTP-mediated destabilization of IL-23 mRNA. A RNA electrophoretic mobility shift assay confirmed that TTP binds to this ARE cluster. Taken together, these results demonstrate that TTP acts as a negative regulator of IL-23 gene expression in mouse colon cancer cells and suggest its potential application as a novel therapeutic target to control IL-23-mediated tumor promotion.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3' Untranslated Regions
  • Animals
  • Binding Sites
  • Cell Line, Tumor
  • Cell Proliferation
  • Colonic Neoplasms / genetics
  • Colonic Neoplasms / metabolism*
  • Colonic Neoplasms / pathology
  • Down-Regulation
  • Gene Expression Regulation, Neoplastic
  • HEK293 Cells
  • Humans
  • Interleukin-23 / genetics*
  • Interleukin-23 / metabolism*
  • Mice
  • Point Mutation
  • RNA Stability
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism*
  • Sequence Deletion
  • Tristetraprolin / genetics
  • Tristetraprolin / metabolism*

Substances

  • 3' Untranslated Regions
  • Interleukin-23
  • RNA, Messenger
  • Tristetraprolin
  • ZFP36 protein, human
  • Zfp36 protein, mouse