Receptors for neuropeptides are induced by exogenous poly(A)+ RNA in oocytes from Xenopus laevis

Proc Natl Acad Sci U S A. 1988 Feb;85(3):714-7. doi: 10.1073/pnas.85.3.714.

Abstract

Receptors for the hormones vasopressin, angiotensin II, and thyrotropin-releasing hormone have been studied electrophysiologically in Xenopus laevis oocytes previously injected with poly(A)+ RNA from the respective receptor-containing tissues. The injected oocytes responded to the hormones by demonstrating oscillations in membrane currents as recorded by the voltage-clamp method. The response was dependent on the hormone concentrations and detectable between 5 and 1000 nM concentrations. Size fractionation of poly(A)+ RNA from the respective tissues showed that the mRNAs encoding the three hormone receptors were larger than 18S rRNA, suggesting a length of at least 2 kilobases. When vasopressin was added to the oocyte bath, an inward membrane current was generated in oocytes injected with rat poly(A)+ RNA from liver but not from kidney. This suggests that the V1-type (liver), not the V2-type (kidney), vasopressin receptor can be expressed and electrophysiologically identified in the oocyte. A V1-specific, but not a V2-specific, antagonist suppressed the vasopressin-dependent effect. Application of angiotensin II to liver poly(A)+ RNA-injected oocytes elicited oscillations in membrane current, indicating that these oocytes also expressed receptors for angiotension II; the antagonist [Sar1, O-methionyl-Tyr4]angiotensin II blocked this effect. Poly(A)+ RNA from tumor-derived GH3B6 cells, known to contain receptors for thyrotropin-releasing hormone, injected into oocytes induced receptors responding to thyrotropin-releasing hormone; the drug chlordiazepoxide suppressed the thyrotropin-releasing hormone response.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Action Potentials / drug effects
  • Angiotensin II / antagonists & inhibitors
  • Angiotensin II / biosynthesis*
  • Angiotensin II / genetics
  • Angiotensin II / pharmacology
  • Angiotensin Receptor Antagonists
  • Animals
  • Female
  • Gene Expression Regulation
  • Ion Channels / drug effects
  • Liver / analysis
  • Multigene Family
  • Oocytes
  • Poly A / biosynthesis
  • Poly A / genetics*
  • RNA, Messenger / biosynthesis
  • RNA, Messenger / genetics*
  • Rats
  • Receptors, Angiotensin / biosynthesis*
  • Receptors, Angiotensin / classification
  • Receptors, Angiotensin / genetics
  • Receptors, Vasopressin
  • Thyrotropin-Releasing Hormone / biosynthesis*
  • Thyrotropin-Releasing Hormone / genetics
  • Thyrotropin-Releasing Hormone / pharmacology
  • Vasopressins / antagonists & inhibitors
  • Vasopressins / pharmacology
  • Xenopus laevis

Substances

  • Angiotensin Receptor Antagonists
  • Ion Channels
  • RNA, Messenger
  • Receptors, Angiotensin
  • Receptors, Vasopressin
  • Vasopressins
  • Angiotensin II
  • Poly A
  • Thyrotropin-Releasing Hormone