A disulphide-linked heterodimer of TWIK-1 and TREK-1 mediates passive conductance in astrocytes

Nat Commun. 2014:5:3227. doi: 10.1038/ncomms4227.

Abstract

TWIK-1 is a member of the two-pore domain K(+) (K2P) channel family that plays an essential part in the regulation of resting membrane potential and cellular excitability. The physiological role of TWIK-1 has remained enigmatic because functional expression of TWIK-1 channels is elusive. Here we report that native TWIK-1 forms a functional channel at the plasma membrane of astrocytes. A search for TWIK-1-binding proteins led to the identification of TREK-1, another member of the K2P family. The TWIK-1/TREK-1 heterodimeric channel is formed via a disulphide bridge between residue C69 in TWIK-1 and C93 in TREK-1. Gene silencing demonstrates that surface expression of TWIK-1 and TREK-1 are interdependent. TWIK-1/TREK-1 heterodimers mediate astrocytic passive conductance and cannabinoid-induced glutamate release from astrocytes. Our study sheds new light on the diversity of K2P channels.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Astrocytes / metabolism*
  • COS Cells
  • Chlorocebus aethiops
  • Dimerization
  • Female
  • Glutamic Acid / metabolism
  • HEK293 Cells
  • Humans
  • Male
  • Mice, Inbred C57BL
  • Potassium / metabolism
  • Potassium Channels, Tandem Pore Domain / metabolism*
  • Receptor, Cannabinoid, CB1

Substances

  • KCNK1 protein, human
  • Potassium Channels, Tandem Pore Domain
  • Receptor, Cannabinoid, CB1
  • potassium channel protein TREK-1
  • Glutamic Acid
  • Potassium