The transcription factor FBI-1 inhibits SAM68-mediated BCL-X alternative splicing and apoptosis

EMBO Rep. 2014 Apr;15(4):419-27. doi: 10.1002/embr.201338241. Epub 2014 Feb 10.

Abstract

Alternative splicing (AS) is tightly coupled to transcription for the majority of human genes. However, how these two processes are linked is not well understood. Here, we unveil a direct role for the transcription factor FBI-1 in the regulation of AS. FBI-1 interacts with the splicing factor SAM68 and reduces its binding to BCL-X mRNA. This, in turn, results in the selection of the proximal 5' splice site in BCL-X exon 2, thereby favoring the anti-apoptotic BCL-XL variant and counteracting SAM68-mediated apoptosis. Conversely, depletion of FBI-1, or expression of a SAM68 mutant lacking the FBI-1 binding region, restores the ability of SAM68 to induce BCL-XS splicing and apoptosis. FBI-1's role in splicing requires the activity of histone deacetylases, whose pharmacological inhibition recapitulates the effects of FBI-1 knockdown. Our study reveals an unexpected function for FBI-1 in splicing modulation with a direct impact on cell survival.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adaptor Proteins, Signal Transducing / physiology*
  • Alternative Splicing*
  • Apoptosis*
  • Cell Line, Tumor
  • DNA-Binding Proteins / physiology*
  • HEK293 Cells
  • Histone Deacetylase 1 / metabolism
  • Humans
  • Protein Binding
  • Protein Interaction Domains and Motifs
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • RNA-Binding Proteins / physiology*
  • Transcription Factors / physiology*
  • Two-Hybrid System Techniques
  • bcl-X Protein / genetics*
  • bcl-X Protein / metabolism

Substances

  • Adaptor Proteins, Signal Transducing
  • DNA-Binding Proteins
  • KHDRBS1 protein, human
  • RNA, Messenger
  • RNA-Binding Proteins
  • Transcription Factors
  • ZBTB7A protein, human
  • bcl-X Protein
  • HDAC1 protein, human
  • Histone Deacetylase 1