Cholecystokinin receptor antagonism of stimulated pancreatic and gastric secretion

J Surg Res. 1989 Nov;47(5):460-4. doi: 10.1016/0022-4804(89)90102-9.

Abstract

The effects of cholecystokinin receptor antagonist, dipentyl-3,4-dichloroproglumide (DDP), on stimulated pancreatic and gastric secretion were studied in the rat. DDP dose-dependently inhibited cholecystokinin-stimulated amylase release from dispersed acinar cells. In vivo, DDP inhibited cholecystokinin octapeptide-stimulated amylase and protein secretion. DDP also inhibited pentagastrin-stimulated gastric acid secretion in vivo. Meal-stimulated acid output was decreased by 34% (DDP 400 micrograms/kg/hr) but responsiveness to histamine or parachlorophenyl-gamma-aminobutyric acid was unchanged.

MeSH terms

  • Amylases / metabolism
  • Animals
  • Food
  • Gastric Acid / metabolism*
  • Kinetics
  • Male
  • Pancreas / drug effects
  • Pancreas / metabolism*
  • Pentagastrin / pharmacology
  • Proglumide / pharmacology
  • Rats
  • Rats, Inbred Strains
  • Receptors, Cholecystokinin / drug effects
  • Receptors, Cholecystokinin / physiology*
  • Sincalide / antagonists & inhibitors
  • Sincalide / pharmacology

Substances

  • Receptors, Cholecystokinin
  • Amylases
  • Pentagastrin
  • Proglumide
  • lorglumide
  • Sincalide