Mustard Gas Inhalation Injury: Therapeutic Strategy

Int J Toxicol. 2014 Jul;33(4):271-281. doi: 10.1177/1091581814532959. Epub 2014 May 6.

Abstract

Mustard gas (sulfur mustard [SM], bis-[2-chloroethyl] sulfide) is a vesicating chemical warfare agent and a potential chemical terrorism agent. Exposure of SM causes debilitating skin blisters (vesication) and injury to the eyes and the respiratory tract; of these, the respiratory injury, if severe, may even be fatal. Therefore, developing an effective therapeutic strategy to protect against SM-induced respiratory injury is an urgent priority of not only the US military but also the civilian antiterrorism agencies, for example, the Homeland Security. Toward developing a respiratory medical countermeasure for SM, four different classes of therapeutic compounds have been evaluated in the past: anti-inflammatory compounds, antioxidants, protease inhibitors and antiapoptotic compounds. This review examines all of these different options; however, it suggests that preventing cell death by inhibiting apoptosis seems to be a compelling strategy but possibly dependent on adjunct therapies using the other drugs, that is, anti-inflammatory, antioxidant, and protease inhibitor compounds.

Keywords: anti-inflammatory; antioxidants; apoptosis; inhalation; protease; sulfur mustard.

Publication types

  • Review
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / therapeutic use*
  • Antidotes / therapeutic use
  • Antioxidants / therapeutic use*
  • Apoptosis / drug effects
  • Chemical Warfare Agents / toxicity*
  • Drug Therapy, Combination
  • Gas Poisoning / drug therapy*
  • Gas Poisoning / immunology
  • Gas Poisoning / metabolism
  • Gas Poisoning / pathology
  • Humans
  • Lung / drug effects
  • Lung / immunology
  • Lung / metabolism
  • Lung / pathology
  • Models, Biological*
  • Mustard Gas / toxicity*
  • Protease Inhibitors / therapeutic use*
  • Respiratory Mucosa / drug effects
  • Respiratory Mucosa / immunology
  • Respiratory Mucosa / metabolism
  • Respiratory Mucosa / pathology

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Antidotes
  • Antioxidants
  • Chemical Warfare Agents
  • Protease Inhibitors
  • Mustard Gas