Stabilization of HAC1 influenza vaccine by spray drying: formulation development and process scale-up

Pharm Res. 2014 Nov;31(11):3006-18. doi: 10.1007/s11095-014-1394-3. Epub 2014 May 24.

Abstract

Purpose: Stable vaccines with long shelf lives and reduced dependency on the cold chain are ideal for stockpiling and rapid deployment during public emergencies, including pandemics. Spray drying is a low-cost process that has potential to produce vaccines stable at a wide range of temperatures. Our aim was to develop a stable formulation of a recombinant H1N1 influenza hemagglutinin vaccine candidate and take it to pilot-scale spray-drying production.

Methods: Eight formulations containing different excipients were produced and assayed for antigen stability, powder characteristics, and immunogenicity after storage at a range of temperatures, resulting in the identification of four promising candidates. A pilot-scale spray-drying process was then developed for further testing of one formulation.

Results: The pilot-scale process was used to reproducibly manufacture three batches of the selected formulation with yields >90%. All batches had stable physical properties and in vitro potency for 6 months at temperatures from -20°C to +50°C. Formulations stored for 3 months elicited immunogenic responses in mice equivalent to a frozen lot of bulk vaccine used as a stability control.

Conclusions: This study demonstrates the feasibility of stabilizing subunit vaccines using a spray-drying process and the suitability of the process for manufacturing a candidate product.

MeSH terms

  • Animals
  • Antigens, Viral / chemistry*
  • Antigens, Viral / immunology
  • Chemistry, Pharmaceutical / methods
  • Drug Stability
  • Drug Storage
  • Excipients / chemistry
  • Hemagglutinin Glycoproteins, Influenza Virus / chemistry*
  • Hemagglutinin Glycoproteins, Influenza Virus / immunology
  • Humans
  • Influenza A Virus, H1N1 Subtype / immunology
  • Influenza Vaccines / chemistry*
  • Influenza Vaccines / immunology
  • Influenza, Human / immunology
  • Mice
  • Mice, Inbred BALB C
  • Powders / chemistry
  • Technology, Pharmaceutical / methods*
  • Temperature

Substances

  • Antigens, Viral
  • Excipients
  • H1N1 virus hemagglutinin
  • Hemagglutinin Glycoproteins, Influenza Virus
  • Influenza Vaccines
  • Powders