Paracrine network: another step in the complexity of resistance to EGFR blockade?

Clin Cancer Res. 2014 Dec 15;20(24):6227-9. doi: 10.1158/1078-0432.CCR-14-1615. Epub 2014 Aug 19.

Abstract

Increased secretion of EGFR ligands amphiregulin and TGFα by limited KRAS-mutant clones is suggested as a paracrine resistance mechanism to anti-EGFR antibodies in colorectal cancer models. These findings are biologically sound but need to be replicated, including in the clinical setting, to foresee whether they are clinically relevant and therapeutically exploitable.

Publication types

  • Comment

MeSH terms

  • Amphiregulin / metabolism*
  • Colorectal Neoplasms / metabolism*
  • Drug Resistance, Neoplasm*
  • ErbB Receptors / antagonists & inhibitors*
  • Humans
  • Paracrine Communication*
  • Transforming Growth Factor alpha / metabolism*

Substances

  • Amphiregulin
  • Transforming Growth Factor alpha
  • ErbB Receptors