Comparison of metabolic effects of aripiprazole, quetiapine and ziprasidone after 12 weeks of treatment in first treated episode of psychosis

Schizophr Res. 2014 Oct;159(1):90-4. doi: 10.1016/j.schres.2014.07.045. Epub 2014 Aug 20.

Abstract

This randomized open-label study compared the incidence of metabolic side effects of aripiprazole, ziprasidone and quetiapine in a population of medication-naïve first-episode psychosis patients. A total of 202 subjects were enrolled. Body weight, body mass index, leptin, fasting lipids and fasting glycaemic parameters were measured at baseline and at 3 months follow-up. A hundred and sixty-six patients completed the follow-up and were included in the analyses. A high proportion of patients experienced a significant weight increase (>7% of their baseline weight): 23% ziprasidone (n=12), 32% with quetiapine (n=16) and 45% with aripiprazole (n=31). Patients treated with aripiprazole gained significantly more weight than the patients in the ziprasidone group (1.2 kg [SD=4.1] versus 4.3 kg [SD=4.8], respectively). The increase in leptin levels was greater in women treated with aripiprazole than in those treated with ziprasidone (p=0.030). Mean prolactin levels significantly increased in patients treated with quetiapine and ziprasidone but not in those treated with aripiprazole. Patients treated with quetiapine and aripiprazole showed a significant increase in total cholesterol and LDL-cholesterol plasma levels. Quetiapine-treated patients resulted in a higher increase in LDL-cholesterol than patients treated with ziprasidone (p=0.021). No other significant differences between groups were found. No significant changes in glycaemic parameters were observed. Our results suggest that ziprasidone has a lower liability for inducing weight gain and lipid abnormalities than aripiprazole or quetiapine.

Keywords: Aripiprazole; First-episode psychosis; Leptin; Medication-naïve; Metabolic side effects; Prolactin; Quetiapine; Weight gain; Ziprasidone.

Publication types

  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Antipsychotic Agents / adverse effects
  • Antipsychotic Agents / therapeutic use*
  • Aripiprazole
  • Cholesterol / blood
  • Dibenzothiazepines / adverse effects
  • Dibenzothiazepines / therapeutic use*
  • Female
  • Follow-Up Studies
  • Humans
  • Male
  • Piperazines / adverse effects
  • Piperazines / therapeutic use*
  • Prolactin / metabolism
  • Psychotic Disorders / drug therapy*
  • Quetiapine Fumarate
  • Quinolones / adverse effects
  • Quinolones / therapeutic use*
  • Sex Factors
  • Thiazoles / adverse effects
  • Thiazoles / therapeutic use*
  • Weight Gain / drug effects

Substances

  • Antipsychotic Agents
  • Dibenzothiazepines
  • Piperazines
  • Quinolones
  • Thiazoles
  • Quetiapine Fumarate
  • ziprasidone
  • Aripiprazole
  • Prolactin
  • Cholesterol