AMP-activated protein kinase activation protects gastric epithelial cells from Helicobacter pylori-induced apoptosis

Biochem Biophys Res Commun. 2014 Oct 10;453(1):13-8. doi: 10.1016/j.bbrc.2014.09.028. Epub 2014 Sep 16.

Abstract

Helicobacter pylori (H pylori), infecting half of the world's population, causes gastritis, duodenal and gastric ulcer, and gastric cancers. AMP-activated protein kinase (AMPK) is a highly conserved regulator of cellular energy and metabolism. Recent studies indicated an important role for AMPK in promoting cell survival. In this study, we discovered that H Pylori induced AMPK activation in transformed (GEC-1 line) and primary human gastric epithelial cells (GECs). Inhibition of H Pylori-stimulated AMPK kinase activity by AMPK inhibitor compound C exacerbated apoptosis in transformed and primary GECs. Meanwhile, downregulation of AMPK expression by targeted shRNAs promoted apoptosis in H pylori-infected GECs. In contrast, A-769662 and resveratrol, two known AMPK activators, or AMPKα1 over-expression, enhanced H Pylori-induced AMPK activation, and inhibited GEC apoptosis. Our data suggested that transforming growth factor-β (TGF-β)-activated kinase 1 (TAK1) could be the upstream kinase for AMPK activation by H pylori. Partial depletion of TAK1 by shRNAs not only inhibited AMPK activation, but also suppressed survival of H pylori-infected GECs. Taken together, these results suggest that TAK1-dependent AMPK activation protects GECs from H pylori-Induced apoptosis.

Keywords: AMPK; Apoptosis; Gastric epithelial cells; Helicobacter pylori; TAK1.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • AMP-Activated Protein Kinases / antagonists & inhibitors
  • AMP-Activated Protein Kinases / genetics
  • AMP-Activated Protein Kinases / metabolism*
  • Apoptosis / drug effects
  • Apoptosis / genetics
  • Apoptosis / physiology*
  • Biphenyl Compounds
  • Cell Line
  • Cell Survival / drug effects
  • Cell Survival / genetics
  • Cell Survival / physiology
  • Cells, Cultured
  • Enzyme Activation / drug effects
  • Epithelial Cells / enzymology
  • Epithelial Cells / microbiology
  • Epithelial Cells / pathology
  • Gastric Mucosa / enzymology*
  • Gastric Mucosa / microbiology*
  • Gastric Mucosa / pathology
  • Gene Expression
  • Helicobacter pylori / pathogenicity*
  • Host-Pathogen Interactions
  • Humans
  • MAP Kinase Kinase Kinases / antagonists & inhibitors
  • MAP Kinase Kinase Kinases / genetics
  • MAP Kinase Kinase Kinases / metabolism
  • Pyrones / pharmacology
  • RNA, Small Interfering / genetics
  • Resveratrol
  • Stilbenes / pharmacology
  • Thiophenes / pharmacology

Substances

  • Biphenyl Compounds
  • Pyrones
  • RNA, Small Interfering
  • Stilbenes
  • Thiophenes
  • MAP Kinase Kinase Kinases
  • MAP kinase kinase kinase 7
  • AMP-Activated Protein Kinases
  • 4-hydroxy-3-(4-(2-hydroxyphenyl)phenyl)-6-oxo-7H-thieno(2,3-b)pyridine-5-carbonitrile
  • Resveratrol