Ferric citrate spans mineral metabolism and anemia domains in ESRD: a review of efficacy and safety data

Expert Rev Clin Pharmacol. 2014 Nov;7(6):705-10. doi: 10.1586/17512433.2014.960848. Epub 2014 Sep 22.

Abstract

Ferric citrate (Zerenex™, Keryx Biopharmaceuticals, Inc.), a phosphate binder drug candidate, recently completed a Phase III program confirming efficacy and demonstrating safety when used to treat hyperphosphatemia in patients with end-stage renal disease. Results of these trials demonstrate that ferric citrate effectively controls serum phosphorus and is well tolerated. Additionally, these studies demonstrate that ferric citrate improves iron parameters and reduces IV iron and erythropoietin stimulating agent utilization while maintaining hemoglobin levels. These unique features may further benefit the management of end-stage renal disease-related anemia.

Keywords: anemia; end-stage renal disease; metabolic bone disease.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Anemia / drug therapy
  • Anemia / etiology
  • Chelating Agents / adverse effects
  • Chelating Agents / pharmacology
  • Chelating Agents / therapeutic use
  • Ferric Compounds / adverse effects
  • Ferric Compounds / pharmacology
  • Ferric Compounds / therapeutic use*
  • Humans
  • Hyperphosphatemia / drug therapy*
  • Hyperphosphatemia / etiology
  • Kidney Failure, Chronic / complications
  • Kidney Failure, Chronic / drug therapy*
  • Phosphates / blood
  • Phosphorus / blood

Substances

  • Chelating Agents
  • Ferric Compounds
  • Phosphates
  • Phosphorus
  • ferric citrate