Mechanism of polyubiquitination by human anaphase-promoting complex: RING repurposing for ubiquitin chain assembly

Mol Cell. 2014 Oct 23;56(2):246-260. doi: 10.1016/j.molcel.2014.09.009. Epub 2014 Oct 9.

Abstract

Polyubiquitination by E2 and E3 enzymes is a predominant mechanism regulating protein function. Some RING E3s, including anaphase-promoting complex/cyclosome (APC), catalyze polyubiquitination by sequential reactions with two different E2s. An initiating E2 ligates ubiquitin to an E3-bound substrate. Another E2 grows a polyubiquitin chain on the ubiquitin-primed substrate through poorly defined mechanisms. Here we show that human APC's RING domain is repurposed for dual functions in polyubiquitination. The canonical RING surface activates an initiating E2-ubiquitin intermediate for substrate modification. However, APC engages and activates its specialized ubiquitin chain-elongating E2 UBE2S in ways that differ from current paradigms. During chain assembly, a distinct APC11 RING surface helps deliver a substrate-linked ubiquitin to accept another ubiquitin from UBE2S. Our data define mechanisms of APC/UBE2S-mediated polyubiquitination, reveal diverse functions of RING E3s and E2s, and provide a framework for understanding distinctive RING E3 features specifying ubiquitin chain elongation.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Apc11 Subunit, Anaphase-Promoting Complex-Cyclosome / metabolism*
  • Apc2 Subunit, Anaphase-Promoting Complex-Cyclosome / metabolism*
  • Apc4 Subunit, Anaphase-Promoting Complex-Cyclosome / metabolism
  • Cell Cycle Checkpoints
  • HeLa Cells
  • Humans
  • Molecular Sequence Data
  • Peptide Biosynthesis, Nucleic Acid-Independent*
  • Polyubiquitin / biosynthesis*
  • Polyubiquitin / genetics
  • Protein Structure, Tertiary
  • Ubiquitin-Conjugating Enzymes / metabolism*
  • Ubiquitination / physiology*

Substances

  • Apc4 Subunit, Anaphase-Promoting Complex-Cyclosome
  • Polyubiquitin
  • Ube2S protein, human
  • Ubiquitin-Conjugating Enzymes
  • Apc11 Subunit, Anaphase-Promoting Complex-Cyclosome
  • Apc2 Subunit, Anaphase-Promoting Complex-Cyclosome

Associated data

  • PDB/2MT5
  • PDB/4R2Y