One-pot synthesis of keto thioethers by palladium/gold-catalyzed click and pinacol reactions

Org Lett. 2014 Nov 7;16(21):5556-9. doi: 10.1021/ol502553p. Epub 2014 Oct 17.

Abstract

An atom-efficient synthesis of keto thioethers was devised via tandem gold/palladium catalysis. The reaction proceeds through a regioselective thiol attack at the β-position of the alcohol, followed by an alkyl, aryl, or benzyl 1,2-shift. Both acyclic and cyclic systems were studied, in the latter case leading to the ring expansion of cyclic substrates.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Benzyl Compounds / chemistry*
  • Catalysis
  • Cyclization
  • Gold / chemistry*
  • Molecular Structure
  • Palladium / chemistry*
  • Sulfides / chemical synthesis*
  • Sulfides / chemistry

Substances

  • Benzyl Compounds
  • Sulfides
  • Palladium
  • Gold