SAH-induced MMP activation and K V current suppression is mediated via both ROS-dependent and ROS-independent mechanisms

Acta Neurochir Suppl. 2015:120:89-94. doi: 10.1007/978-3-319-04981-6_15.

Abstract

Voltage-gated potassium (K V) channels regulate cerebral artery tone and have been implicated in subarachnoid hemorrhage (SAH)-induced pathologies. Here, we examined whether matrix metalloprotease (MMP) activation contributes to SAH-induced K V current suppression and cerebral artery constriction via activation of epidermal growth factor receptors (EGFRs). Using patch clamp electrophysiology, we observed that K V currents were selectively decreased in cerebral artery myocytes isolated from SAH model rabbits. Consistent with involvement of enhanced MMP and EGFR activity in SAH-induced K V current suppression, we found that: (1) oxyhemoglobin (OxyHb) and/or the exogenous EGFR ligand, heparin-binding EGF-like growth factor (HB-EGF), failed to induce further K V current suppression after SAH and (2) gelatin zymography detected significantly higher MMP-2 activity after SAH. The removal of reactive oxygen species (ROS) by combined treatment with superoxide dismutase (SOD) and catalase partially inhibited OxyHb-induced K V current suppression. However, these agents had little effect on OxyHb-induced MMP-2 activation. Interestingly, in the presence of a broad-spectrum MMP inhibitor (GM6001), OxyHb failed to cause K V current suppression. These data suggest that OxyHb suppresses K V currents through both ROS-dependent and ROS-independent pathways involving MMP activation. The ROS-independent pathway involves activation of MMP-2, whereas the ROS-dependent pathway involves activation of a second unidentified MMP or ADAM (a disintegrin and metalloprotease domain).

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Dipeptides / pharmacology
  • Disease Models, Animal
  • ErbB Receptors / metabolism
  • Heparin-binding EGF-like Growth Factor / metabolism
  • Heparin-binding EGF-like Growth Factor / pharmacology
  • Matrix Metalloproteinase 2 / metabolism*
  • Matrix Metalloproteinase Inhibitors / pharmacology
  • Oxyhemoglobins / metabolism
  • Patch-Clamp Techniques
  • Potassium Channels, Voltage-Gated / physiology*
  • Rabbits
  • Reactive Oxygen Species / metabolism*
  • Subarachnoid Hemorrhage / drug therapy
  • Subarachnoid Hemorrhage / metabolism*
  • Subarachnoid Hemorrhage / physiopathology*

Substances

  • Dipeptides
  • Heparin-binding EGF-like Growth Factor
  • Matrix Metalloproteinase Inhibitors
  • N-(2(R)-2-(hydroxamidocarbonylmethyl)-4-methylpentanoyl)-L-tryptophan methylamide
  • Oxyhemoglobins
  • Potassium Channels, Voltage-Gated
  • Reactive Oxygen Species
  • ErbB Receptors
  • Matrix Metalloproteinase 2