A positive role of DBC1 in PEA3-mediated progression of estrogen receptor-negative breast cancer

Oncogene. 2015 Aug 20;34(34):4500-8. doi: 10.1038/onc.2014.381. Epub 2014 Nov 24.

Abstract

Deleted in Breast Cancer 1 (DBC1), a negative regulator of deacetylase SIRT1, has been shown to act as an estrogen receptor α (ER) coactivator that has a key role in ER transcription complex assembly and estrogen-dependent breast cancer cell proliferation. However, little is known about its physiological role and mechanism of action in ER-negative breast cancer cells. Here we report that DBC1 functions as a coactivator for the oncogenic ETS transcription factor PEA3 to promote ER-negative breast cancer progression. DBC1 is required for the expression of PEA3 target genes and for recruitment of PEA3 and RNA polymerase II to PEA3 target promoters. We also demonstrated that acetylation of PEA3 stimulates its DNA binding and association with DBC1 by disrupting the intramolecular interaction of PEA3. The molecular mechanism underlying DBC1 function in PEA3-mediated transcription involves inhibition of SIRT1 interaction with PEA3 and of SIRT1-mediated deacetylation of PEA3. Moreover, DBC1 depletion inhibited the tumorigenic properties of ER-negative breast cancer cells in vitro and in vivo. Importantly, increased DBC1 expression correlated with shorter relapse-free survival of ER-negative breast cancer patients. Our results firmly established DBC1 as a critical coactivator of PEA3 and as a key player in PEA3-mediated breast cancer progression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylation
  • Adaptor Proteins, Signal Transducing / chemistry
  • Adaptor Proteins, Signal Transducing / physiology*
  • Adenovirus E1A Proteins / physiology*
  • Binding Sites
  • Breast Neoplasms / chemistry
  • Breast Neoplasms / etiology*
  • Cell Line, Tumor
  • Disease Progression
  • Female
  • Humans
  • Protein Conformation
  • Proto-Oncogene Proteins / physiology*
  • Proto-Oncogene Proteins c-ets
  • Receptors, Estrogen / analysis*
  • Sirtuin 1 / physiology

Substances

  • Adaptor Proteins, Signal Transducing
  • Adenovirus E1A Proteins
  • CCAR2 protein, human
  • ETV4 protein, human
  • Proto-Oncogene Proteins
  • Proto-Oncogene Proteins c-ets
  • Receptors, Estrogen
  • SIRT1 protein, human
  • Sirtuin 1