Blocking lymphocyte trafficking with FTY720 prevents inflammation-sensitized hypoxic-ischemic brain injury in newborns

J Neurosci. 2014 Dec 3;34(49):16467-81. doi: 10.1523/JNEUROSCI.2582-14.2014.

Abstract

Intrauterine infection (chorioamnionitis) aggravates neonatal hypoxic-ischemic (HI) brain injury, but the mechanisms linking systemic inflammation to the CNS damage remain uncertain. Here we report evidence for brain influx of T-helper 17 (TH17)-like lymphocytes to coordinate neuroinflammatory responses in lipopolysaccharide (LPS)-sensitized HI injury in neonates. We found that both infants with histological chorioamnionitis and rat pups challenged by LPS/HI have elevated expression of the interleukin-23 (IL-23) receptor, a marker of early TH17 lymphocytes, in the peripheral blood mononuclear cells. Post-LPS/HI administration of FTY720 (fingolimod), a sphingosine-1-phosphate receptor agonist that blocks lymphocyte trafficking, mitigated the influx of leukocytes through the choroid plexus and acute induction of nuclear factor-κB signaling in the brain. Subsequently, the FTY720 treatment led to attenuated blood-brain barrier damage, fewer cluster of differentiation 4-positive, IL-17A-positive T-cells in the brain, less proinflammatory cytokine, and better preservation of growth and white matter functions. The FTY720 treatment also provided dose-dependent reduction of brain atrophy, rescuing >90% of LPS/HI-induced brain tissue loss. Interestingly, FTY720 neither opposed pure-HI brain injury nor directly inhibited microglia in both in vivo and in vitro models, highlighting its unique mechanism against inflammation-sensitized HI injury. Together, these results suggest that the dual hit of systemic inflammation and neonatal HI injury triggers early onset of the TH17/IL-17-mediated immunity, which causes severe brain destruction but responds remarkably to the therapeutic blockade of lymphocyte trafficking.

Keywords: FTY720; Fingolimod; Th17; adaptive immunity; chorioamnionitis; choroid plexus.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Animals, Newborn
  • Atrophy / drug therapy
  • Blood-Brain Barrier / drug effects
  • Brain / drug effects
  • Brain / metabolism
  • Brain / pathology
  • Cell Movement / drug effects*
  • Chorioamnionitis / drug therapy
  • Chorioamnionitis / metabolism
  • Cytokines / metabolism
  • Dose-Response Relationship, Drug
  • Female
  • Fingolimod Hydrochloride
  • Humans
  • Hypoxia-Ischemia, Brain / drug therapy
  • Hypoxia-Ischemia, Brain / pathology*
  • Hypoxia-Ischemia, Brain / prevention & control*
  • Immunosuppressive Agents / pharmacology
  • Immunosuppressive Agents / therapeutic use
  • Infant, Newborn
  • Inflammation / prevention & control*
  • Lipopolysaccharides
  • Lymphocyte Activation / drug effects*
  • Lymphocytes / cytology
  • Lymphocytes / drug effects*
  • NF-kappa B / metabolism
  • Pregnancy
  • Propylene Glycols / pharmacology*
  • Propylene Glycols / therapeutic use
  • Rats
  • Receptors, Interleukin / metabolism
  • Sphingosine / analogs & derivatives*
  • Sphingosine / pharmacology
  • Sphingosine / therapeutic use
  • T-Lymphocytes / cytology
  • T-Lymphocytes / drug effects
  • White Matter / drug effects

Substances

  • Cytokines
  • IL23R protein, human
  • Immunosuppressive Agents
  • Lipopolysaccharides
  • NF-kappa B
  • Propylene Glycols
  • Receptors, Interleukin
  • Fingolimod Hydrochloride
  • Sphingosine