Muscarinic acetylcholine receptor M3 modulates odorant receptor activity via inhibition of β-arrestin-2 recruitment

Nat Commun. 2015 Mar 24:6:6448. doi: 10.1038/ncomms7448.

Abstract

The olfactory system in rodents serves a critical function in social, reproductive and survival behaviours. Processing of chemosensory signals in the brain is dynamically regulated in part by an animal's physiological state. We previously reported that type 3 muscarinic acetylcholine receptors (M3-Rs) physically interact with odorant receptors (ORs) to promote odour-induced responses in a heterologous expression system. However, it is not known how M3-Rs affect the ability of olfactory sensory neurons (OSNs) to respond to odours. Here, we show that an M3-R antagonist attenuates odour-induced responses in OSNs from wild-type, but not M3-R-null, mice. Using a novel molecular assay, we demonstrate that the activation of M3-Rs inhibits the recruitment of β-arrestin-2 to ORs, resulting in a potentiation of odour-induced responses in OSNs. These results suggest a role for acetylcholine in modulating olfactory processing at the initial stages of signal transduction in the olfactory system.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Arrestins / drug effects
  • Arrestins / genetics*
  • Arrestins / metabolism
  • Benzofurans / pharmacology
  • Calcium Signaling
  • Cyclic AMP / metabolism
  • HEK293 Cells
  • Humans
  • Immunohistochemistry
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Muscarinic Antagonists / pharmacology
  • Odorants
  • Olfactory Receptor Neurons
  • Patch-Clamp Techniques
  • Pyrrolidines / pharmacology
  • Receptor, Muscarinic M3 / antagonists & inhibitors
  • Receptor, Muscarinic M3 / genetics*
  • Receptor, Muscarinic M3 / metabolism
  • Receptors, Odorant / drug effects
  • Receptors, Odorant / metabolism*
  • Type C Phospholipases / metabolism
  • beta-Arrestin 2
  • beta-Arrestins

Substances

  • ARRB2 protein, human
  • Arrb2 protein, mouse
  • Arrestins
  • Benzofurans
  • Muscarinic Antagonists
  • Pyrrolidines
  • Receptor, Muscarinic M3
  • Receptors, Odorant
  • beta-Arrestin 2
  • beta-Arrestins
  • darifenacin
  • Cyclic AMP
  • Type C Phospholipases