Bcl-xL stimulates Bax relocation to mitochondria and primes cells to ABT-737

Int J Biochem Cell Biol. 2015 Jul:64:136-46. doi: 10.1016/j.biocel.2015.03.020. Epub 2015 Apr 8.

Abstract

Bax cytosol-to-mitochondria translocation is a central event of the intrinsic pathway of apoptosis. Bcl-xL is an important regulator of this event and was recently shown to promote the retrotranslocation of mitochondrial Bax to the cytosol. The present study identifies a new aspect of the regulation of Bax localization by Bcl-xL: in addition to its role in Bax inhibition and retrotranslocation, we found that, like with Bcl-2, an increase of Bcl-xL expression levels led to an increase of Bax mitochondrial content. This finding was substantiated both in pro-lymphocytic FL5.12 cells and a yeast reporting system. Bcl-xL-dependent increase of mitochondrial Bax is counterbalanced by retrotranslocation, as we observed that Bcl-xLΔC, which is unable to promote Bax retrotranslocation, was more efficient than the full-length protein in stimulating Bax relocation to mitochondria. Interestingly, cells overexpressing Bcl-xL were more sensitive to apoptosis upon treatment with the BH3-mimetic ABT-737, suggesting that despite its role in Bax inhibition, Bcl-xL also primes mitochondria to permeabilization and cytochrome c release.

Keywords: Apoptosis; BH3-mimetics; Bcl-2 family; Mitochondria.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / pharmacology*
  • Apoptosis
  • Biphenyl Compounds / pharmacology*
  • Cell Line
  • Mice
  • Mitochondria / metabolism*
  • Nitrophenols / pharmacology*
  • Piperazines / pharmacology
  • Protein Multimerization
  • Protein Transport
  • Saccharomyces cerevisiae
  • Sulfonamides / pharmacology*
  • bcl-2-Associated X Protein / metabolism*
  • bcl-X Protein / metabolism*

Substances

  • ABT-737
  • Antineoplastic Agents
  • Bax protein, mouse
  • Bcl2l1 protein, mouse
  • Biphenyl Compounds
  • Nitrophenols
  • Piperazines
  • Sulfonamides
  • bcl-2-Associated X Protein
  • bcl-X Protein