Improvement of bone marrow fibrosis with ruxolitinib: will this finding change our perception of the drug?

Expert Rev Hematol. 2015 Aug;8(4):387-9. doi: 10.1586/17474086.2015.1041494. Epub 2015 Apr 27.

Abstract

Ruxolitinib, a JAK1 and JAK2 inhibitor, has been tested and approved for the treatment of primary and secondary myelofibrosis. Reduction of spleen volume and improvement of constitutional symptoms and quality of life have been reported as the major findings in sponsored randomized clinical trials. Recent data indicated that the drug improves bone marrow fibrosis and that different targets may be involved in this response. These new data, which require confirmation in prospective trials, may change our perspectives and therapeutic strategies for this disease.

Keywords: fibrosis; myelofibrosis; ruxolitinib.

Publication types

  • Editorial

MeSH terms

  • Humans
  • Janus Kinases / antagonists & inhibitors
  • Nitriles
  • Primary Myelofibrosis / drug therapy*
  • Primary Myelofibrosis / metabolism
  • Protein Kinase Inhibitors / pharmacology
  • Protein Kinase Inhibitors / therapeutic use*
  • Pyrazoles / pharmacology
  • Pyrazoles / therapeutic use*
  • Pyrimidines
  • Treatment Outcome

Substances

  • Nitriles
  • Protein Kinase Inhibitors
  • Pyrazoles
  • Pyrimidines
  • ruxolitinib
  • Janus Kinases