The role of denosumab in the prevention of hypercalcaemia of malignancy in cancer patients with metastatic bone disease

Eur J Cancer. 2015 Jul;51(11):1467-75. doi: 10.1016/j.ejca.2015.04.017. Epub 2015 May 11.

Abstract

Background: We compared the activity of denosumab with zoledronic acid for delaying or preventing hypercalcaemia of malignancy (HCM) in patients with advanced cancer and bone metastases or with multiple myeloma.

Methods: Patient-level data were combined from two identically designed, randomised, double-blind, active-controlled, phase III trials of advanced cancer patients with breast cancer and other solid tumours (excluding breast or prostate cancer) or multiple myeloma. End-points included time to first on-study HCM, time to first and subsequent on-study HCM, proportion of patients experiencing HCM and proportion of patients experiencing recurrent HCM.

Results: Denosumab significantly delayed the time to first on-study HCM, representing a 37% reduction in the hazard ratio (HR) compared with zoledronic acid (HR, 0.63; 95% confidence interval (CI): 0.41-0.98; P = 0.042) and reduced the risk of developing recurrent HCM (time to first and subsequent on-study HCM) by 52% (rate ratio, 0.48; 95% CI: 0.29-0.81; P = 0.006). The median time on study was 12.9 months. Fewer patients receiving denosumab compared with zoledronic acid experienced an HCM event (1.7% versus 2.7%; P = 0.028). Of the 84 patients experiencing an HCM event, 40% of those receiving zoledronic acid experienced >1 event of HCM compared with 31% of those receiving denosumab.

Conclusion: Denosumab treatment was more efficacious than treatment with zoledronic acid in delaying or preventing HCM in advanced cancer patients with breast cancer, other solid tumours or multiple myeloma.

Trial registration: ClinicalTrials.gov NCT00321464 NCT00330759.

Keywords: Breast cancer; Denosumab; Hypercalcaemia of malignancy; Multiple myeloma; Solid tumours; Supportive care; Zoledronic acid.

Publication types

  • Clinical Trial, Phase III
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antibodies, Monoclonal, Humanized / therapeutic use*
  • Bone Neoplasms / blood*
  • Bone Neoplasms / secondary*
  • Breast Neoplasms / blood
  • Breast Neoplasms / pathology
  • Denosumab
  • Diphosphonates / therapeutic use
  • Double-Blind Method
  • Female
  • Humans
  • Hypercalcemia / prevention & control*
  • Imidazoles / therapeutic use
  • Male
  • Middle Aged
  • Multiple Myeloma / blood
  • Multiple Myeloma / pathology
  • Neoplasms / blood*
  • Neoplasms / pathology*
  • Proportional Hazards Models
  • Zoledronic Acid

Substances

  • Antibodies, Monoclonal, Humanized
  • Diphosphonates
  • Imidazoles
  • Denosumab
  • Zoledronic Acid

Associated data

  • ClinicalTrials.gov/NCT00321464
  • ClinicalTrials.gov/NCT00330759