NF-κB decoy oligodeoxynucleotide inhibits wear particle-induced inflammation in a murine calvarial model

J Biomed Mater Res A. 2015 Dec;103(12):3872-8. doi: 10.1002/jbm.a.35532. Epub 2015 Jul 14.

Abstract

Wear particles induce periprosthetic inflammation and osteolysis through activation of nuclear factor kappa B (NF-κB), which up-regulates the downstream target gene expression for proinflammatory cytokines in macrophages. It was hypothesized that direct suppression of NF-κB activity in the early phases of this disorder could be a therapeutic strategy for preventing the inflammatory response to wear particles, potentially mitigating osteolysis. NF-κB activity can be suppressed via competitive binding with double stranded NF-κB decoy oligodeoxynucleotides (ODNs) that blocks this transcription factor from binding to the promoter regions of targeted genes. In this murine calvarial study, clinically relevant polyethylene particles (PEs) with/without ODN were subcutaneously injected over the calvarial bone. In the presence of PE particles, macrophages migrated to the inflammatory site and induced tumor necrosis factor alpha (TNF-α) and receptor activator of nuclear factor kappa B ligand (RANKL) expression, resulting in an increase in the number of osteoclasts. Local injections of ODN mitigated the expression of TNF-α, RANKL, and induced the expression of two anti-inflammatory, antiresorptive cytokines: interleukin-1 receptor antagonist and osteoprotegerin. Local intervention with NF-κB decoy ODN in early cases of particle-induced inflammation in which the prosthesis is still salvageable may potentially preserve periprosthetic bone stock.

Keywords: NF-κB; murine calvarial model; osteolysis; total joint replacement; wear particles.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Inflammation / drug therapy*
  • Inflammation / immunology*
  • Inflammation / pathology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • NF-kappa B
  • Oligodeoxyribonucleotides / therapeutic use*
  • Organ Culture Techniques
  • Particle Size
  • Polyethylene / analysis
  • Polyethylene / immunology*
  • Skull / drug effects*
  • Skull / immunology*
  • Skull / pathology

Substances

  • NF-kappa B
  • NF-kappaB decoy
  • Oligodeoxyribonucleotides
  • Polyethylene