COP9 signalosome subunit 6 (CSN6) regulates E6AP/UBE3A in cervical cancer

Oncotarget. 2015 Sep 29;6(29):28026-41. doi: 10.18632/oncotarget.4731.

Abstract

Cervical cancer is one of the leading causes of cancer death in women. Human papillomaviruses (HPVs) are the major cause in almost 99.7% of cervical cancer. E6 oncoprotein of HPV and E6-associated protein (E6AP) are critical in causing p53 degradation and malignancy. Understanding the E6AP regulation is critical to develop treating strategy for cervical cancer patients. The COP9 signalosome subunit 6 (CSN6) is involved in ubiquitin-mediated protein degradation. We found that both CSN6 and E6AP are overexpressed in cervical cancer. We characterized that CSN6 associated with E6AP and stabilized E6AP expression by reducing E6AP poly-ubiquitination, thereby regulating p53 activity in cell proliferation and apoptosis. Mechanistic studies revealed that CSN6-E6AP axis can be regulated by EGF/Akt signaling. Furthermore, inhibition of CSN6-E6AP axis hinders cervical cancer growth in mice. Taken together, our results indicate that CSN6 is a positive regulator of E6AP and is important for cervical cancer development.

Keywords: CSN6; E6AP; cervical cancer; p53; ubiquitination.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Adaptor Proteins, Signal Transducing / metabolism*
  • Animals
  • COP9 Signalosome Complex
  • Cell Separation
  • Cell Transformation, Neoplastic / genetics
  • Female
  • Flow Cytometry
  • Gene Expression Regulation, Neoplastic / genetics*
  • HeLa Cells
  • Humans
  • Immunoblotting
  • Immunoprecipitation
  • Mice
  • Mice, Nude
  • Papillomavirus Infections / complications*
  • Polymerase Chain Reaction
  • RNA, Small Interfering
  • Transfection
  • Ubiquitin-Protein Ligases / metabolism*
  • Uterine Cervical Neoplasms / genetics*
  • Uterine Cervical Neoplasms / pathology*
  • Uterine Cervical Neoplasms / virology
  • Xenograft Model Antitumor Assays

Substances

  • Adaptor Proteins, Signal Transducing
  • COPS6 protein, human
  • RNA, Small Interfering
  • UBE3A protein, human
  • Ubiquitin-Protein Ligases
  • COP9 Signalosome Complex