Pharmacokinetics of 99mTc-MAA- and 99mTc-HSA-Microspheres Used in Preradioembolization Dosimetry: Influence on the Liver-Lung Shunt

J Nucl Med. 2016 Jun;57(6):925-7. doi: 10.2967/jnumed.115.169987. Epub 2016 Feb 9.

Abstract

Perfusion scintigraphy using (99m)Tc-labeled albumin aggregates is mandatory before hepatic radioembolization with (90)Y-microspheres. As part of a prospective trial, the intrahepatic and intrapulmonary stability of 2 albumin compounds, (99m)Tc-MAA (macroaggregated serum albumin [MAA]) and (99m)Tc-HSA (human serum albumin [HSA]), was assessed.

Methods: In 24 patients with metastatic colorectal cancer, biodistribution (liver, lung) and liver-lung shunt (LLS) of both tracers (12 patients each) were assessed by sequential planar scintigraphy (1, 5, and 24 h after injection).

Results: Liver uptake of both albumin compounds decreased differently. Although initial LLSs at 1 h after injection were similar in both groups, MAA-LLS increased significantly from 1 (3.9%) to 5 h (7.7%) and 24 h (9.9%) after injection, respectively. HSA-LLS did not change significantly (1 to 5 h), indicating a steady state of pulmonary and intrahepatic degradation.

Conclusion: Compared with (99m)Tc-MAA-microspheres, (99m)Tc-HSA-microspheres are likely more resistant to degradation over time, allowing a reliable LLS determination even at later time points.

Keywords: 99mTc-labeled albumin spheres; biokinetics; dosimetry; liver-lung shunt; radioembolization.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Aged
  • Aged, 80 and over
  • Colorectal Neoplasms / pathology
  • Embolization, Therapeutic*
  • Female
  • Humans
  • Liver / diagnostic imaging
  • Liver / metabolism*
  • Liver / radiation effects
  • Liver Neoplasms / diagnostic imaging
  • Liver Neoplasms / metabolism
  • Liver Neoplasms / radiotherapy
  • Liver Neoplasms / secondary
  • Lung / diagnostic imaging
  • Lung / metabolism*
  • Lung / radiation effects
  • Male
  • Microspheres*
  • Middle Aged
  • Perfusion Imaging
  • Prospective Studies
  • Technetium Tc 99m Aggregated Albumin / chemistry*
  • Technetium Tc 99m Aggregated Albumin / pharmacokinetics*
  • Tissue Distribution

Substances

  • Technetium Tc 99m Aggregated Albumin