Myoscape controls cardiac calcium cycling and contractility via regulation of L-type calcium channel surface expression

Nat Commun. 2016 Apr 28:7:11317. doi: 10.1315/11317.

Abstract

Calcium signalling plays a critical role in the pathogenesis of heart failure. Here we describe a cardiac protein named Myoscape/FAM40B/STRIP2, which directly interacts with the L-type calcium channel. Knockdown of Myoscape in cardiomyocytes decreases calcium transients associated with smaller Ca(2+) amplitudes and a lower diastolic Ca(2+) content. Likewise, L-type calcium channel currents are significantly diminished on Myoscape ablation, and downregulation of Myoscape significantly reduces contractility of cardiomyocytes. Conversely, overexpression of Myoscape increases global Ca(2+) transients and enhances L-type Ca(2+) channel currents, and is sufficient to restore decreased currents in failing cardiomyocytes. In vivo, both Myoscape-depleted morphant zebrafish and Myoscape knockout (KO) mice display impairment of cardiac function progressing to advanced heart failure. Mechanistically, Myoscape-deficient mice show reduced L-type Ca(2+)currents, cell capacity and calcium current densities as a result of diminished LTCC surface expression. Finally, Myoscape expression is reduced in hearts from patients suffering of terminal heart failure, implying a role in human disease.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Animals, Newborn
  • Calcium / metabolism*
  • Calcium Channels, L-Type / genetics*
  • Calcium Channels, L-Type / metabolism
  • Carrier Proteins / genetics*
  • Carrier Proteins / metabolism
  • Cells, Cultured
  • Cytoskeletal Proteins
  • Gene Expression Regulation*
  • HEK293 Cells
  • Humans
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Myocardial Contraction / genetics
  • Myocardium / metabolism*
  • Myocytes, Cardiac / cytology
  • Myocytes, Cardiac / metabolism
  • Myocytes, Cardiac / physiology
  • Protein Binding
  • Rats, Sprague-Dawley
  • Rats, Wistar
  • Zebrafish / genetics
  • Zebrafish / metabolism

Substances

  • CACNA1C protein, human
  • Calcium Channels, L-Type
  • Carrier Proteins
  • Cytoskeletal Proteins
  • STRIP2 protein, human
  • Calcium