The Effect of Latency Reversal Agents on Primary CD8+ T Cells: Implications for Shock and Kill Strategies for Human Immunodeficiency Virus Eradication

EBioMedicine. 2016 Jun:8:217-229. doi: 10.1016/j.ebiom.2016.04.019. Epub 2016 Apr 18.

Abstract

Shock and kill strategies involving the use of small molecules to induce viral transcription in resting CD4+ T cells (shock) followed by immune mediated clearance of the reactivated cells (kill), have been proposed as a method of eliminating latently infected CD4+ T cells. The combination of the histone deacetylase (HDAC) inhibitor romidepsin and protein kinase C (PKC) agonist bryostatin-1 is very effective at reversing latency in vitro. However, we found that primary HIV-1 specific CD8+ T cells were not able to eliminate autologous resting CD4+ T cells that had been reactivated with these drugs. We tested the hypothesis that the drugs affected primary CD8+ T cell function and found that both agents had inhibitory effects on the suppressive capacity of HIV-specific CD8+ T cells from patients who control viral replication without antiretroviral therapy (elite suppressors/controllers). The inhibitory effect was additive and multi-factorial in nature. These inhibitory effects were not seen with prostratin, another PKC agonist, either alone or in combination with JQ1, a bromodomain-containing protein 4 inhibitor. Our results suggest that because of their adverse effects on primary CD8+ T cells, some LRAs may cause immune-suppression and therefore should be used with caution in shock and kill strategies.

Keywords: CD8+ T cells; Elite controllers; Elite suppressors; Eradication; HIV-1; Latency reversal agents.

MeSH terms

  • Antiretroviral Therapy, Highly Active
  • Biomarkers
  • Bryostatins / pharmacology
  • CD4 Lymphocyte Count
  • CD4-Positive T-Lymphocytes / drug effects
  • CD4-Positive T-Lymphocytes / immunology
  • CD4-Positive T-Lymphocytes / metabolism
  • CD4-Positive T-Lymphocytes / virology
  • CD8-Positive T-Lymphocytes / drug effects
  • CD8-Positive T-Lymphocytes / immunology*
  • CD8-Positive T-Lymphocytes / metabolism
  • Cytokines / metabolism
  • Depsipeptides / pharmacology
  • Female
  • HIV Infections / drug therapy
  • HIV Infections / immunology*
  • HIV Infections / virology*
  • HIV-1 / physiology*
  • HLA-A Antigens / immunology
  • HLA-B Antigens / immunology
  • Humans
  • Immunomodulation / drug effects
  • Lymphocyte Activation / immunology
  • Male
  • Receptors, Antigen, T-Cell / metabolism
  • Viral Load
  • Virus Activation
  • Virus Latency*

Substances

  • Biomarkers
  • Bryostatins
  • Cytokines
  • Depsipeptides
  • HLA-A Antigens
  • HLA-B Antigens
  • Receptors, Antigen, T-Cell
  • bryostatin 1
  • romidepsin