Abstract
Oncogenic fusions in TRK family receptor tyrosine kinases have been identified in several cancers and can serve as therapeutic targets. We identified ETV6-NTRK3, MYO5A-NTRK3 and MYH9-NTRK3 fusions in Spitz tumours, and demonstrated that NTRK3 fusions constitutively activate the mitogen-activated protein kinase, phosphoinositide 3-kinase and phospholipase Cγ1 pathways in melanocytes. This signalling was inhibited by DS-6051a, a small-molecule inhibitor of NTRK1/2/3 and ROS1. NTRK3 fusions expand the range of oncogenic kinase fusions in melanocytic neoplasms and offer targets for a small subset of melanomas for which no targeted options currently exist. Copyright © 2016 Pathological Society of Great Britain and Ireland. Published by John Wiley & Sons, Ltd.
Keywords:
NTRK3 fusion; Spitz naevus; Spitz tumour; atypical Spitz tumour; genetics; kinase inhibitor; melanoma; oncogene; spitzoid melanoma.
Copyright © 2016 Pathological Society of Great Britain and Ireland. Published by John Wiley & Sons, Ltd.
Publication types
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Research Support, N.I.H., Extramural
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Research Support, Non-U.S. Gov't
MeSH terms
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Adolescent
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Adult
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Aged
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Child
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Child, Preschool
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Comparative Genomic Hybridization
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Discoidin Domain Receptor 2 / genetics*
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Discoidin Domain Receptor 2 / metabolism
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ETS Translocation Variant 6 Protein
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Female
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Humans
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Male
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Melanoma / enzymology
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Melanoma / genetics
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Melanoma / pathology
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Mitogen-Activated Protein Kinases / genetics
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Mitogen-Activated Protein Kinases / metabolism
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Molecular Motor Proteins / genetics*
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Molecular Motor Proteins / metabolism
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Myosin Heavy Chains / genetics*
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Myosin Heavy Chains / metabolism
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Myosin Type V / genetics*
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Myosin Type V / metabolism
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Nevus, Epithelioid and Spindle Cell / enzymology*
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Nevus, Epithelioid and Spindle Cell / genetics
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Nevus, Epithelioid and Spindle Cell / pathology
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Oncogene Fusion
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Phosphatidylinositol 3-Kinases / genetics
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Phosphatidylinositol 3-Kinases / metabolism
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Proto-Oncogene Proteins c-ets / genetics*
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Proto-Oncogene Proteins c-ets / metabolism
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Repressor Proteins / genetics*
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Repressor Proteins / metabolism
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Sequence Analysis, DNA
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Sequence Analysis, RNA
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Skin Neoplasms / enzymology*
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Skin Neoplasms / genetics
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Skin Neoplasms / pathology
Substances
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MYH9 protein, human
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Molecular Motor Proteins
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Proto-Oncogene Proteins c-ets
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Repressor Proteins
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MYO5A protein, human
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Phosphatidylinositol 3-Kinases
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DDR2 protein, human
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Discoidin Domain Receptor 2
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Mitogen-Activated Protein Kinases
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Myosin Type V
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Myosin Heavy Chains