TEA prevents inactivation while blocking open K+ channels in human T lymphocytes

Biophys J. 1989 Jan;55(1):203-6. doi: 10.1016/S0006-3495(89)82793-6.

Abstract

The whole-cell recording mode of the patch-clamp technique was used to study the effect of external tetraethylammonium ([TEA+]o) on the inactivating, voltage-dependent K+ channels of human T lymphocytes. TEA+ reduced the peak amplitude and slowed the time course of the K+ current decay during a depolarizing pulse, resulting in a crossover of the current records in the presence and absence of TEA+. In solutions with different [TEA+]o both the peak K+ current amplitude, lKpeak, and the time constant of the decay of the K+ current, tau d, were reduced in a dose-dependent manner, both with apparent binding constants, KD, of 12 mM. The integral of K+ current during a prolonged depolarizing pulse was unaltered in solutions with different [TEA+]o. The concentration dependence of [TEA+]o on lKpeak, tau d, and the unchanged current integral can be explained with a kinetic scheme in which open channels blocked by TEA+ cannot inactivate.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Cell Line
  • Electrophysiology / methods
  • Humans
  • Kinetics
  • Mathematics
  • Membrane Potentials
  • Models, Theoretical
  • Potassium Channels / drug effects
  • Potassium Channels / physiology*
  • T-Lymphocytes / drug effects
  • T-Lymphocytes / physiology*
  • Tetraethylammonium
  • Tetraethylammonium Compounds / pharmacology*

Substances

  • Potassium Channels
  • Tetraethylammonium Compounds
  • Tetraethylammonium