Sexual Reassignment Fails to Prevent Kennedy's Disease

J Neuromuscul Dis. 2016 Mar 3;3(1):121-125. doi: 10.3233/JND-150128.

Abstract

Spinal and bulbar muscular atrophy is caused by polyglutamine expansion in the androgen receptor. As an X-linked disease dependent on androgens, symptoms and findings are only fully manifest in males. Here we describe a 40-year-old male-to-female transgender SBMA patient who developed full disease manifestations despite undetectable levels of androgens. We used cell culture and animal models to show that spironolactone, the anti-androgen she had taken for 15 years, promotes nuclear localization and toxicity of the mutant protein, which may explain the disease manifestations in this patient.

Keywords: Motor neuron disease; X-Linked; androgen; bulbo-spinal atrophy; receptors; spironolactone.

Publication types

  • Case Reports

MeSH terms

  • Androgen Antagonists / adverse effects
  • Androgen Antagonists / pharmacology*
  • Animals
  • Bulbo-Spinal Atrophy, X-Linked / prevention & control*
  • Disease Models, Animal
  • Drosophila
  • Female
  • Humans
  • Male
  • Rats
  • Sex Reassignment Procedures / methods*
  • Spironolactone / adverse effects
  • Spironolactone / pharmacology*
  • Transsexualism / therapy*

Substances

  • Androgen Antagonists
  • Spironolactone