Resveratrol Inhibited Non-small Cell Lung Cancer Through Inhibiting STAT-3 Signaling

Am J Med Sci. 2016 Nov;352(5):524-530. doi: 10.1016/j.amjms.2016.08.027. Epub 2016 Sep 22.

Abstract

Background: Resveratrol has demonstrated many beneficial effects against cancers; however, the mechanism remains unclear. Non-small cell lung cancer accounts for 80% of lung cancers. The present study was designed to observe the effects and related mechanisms of resveratrol on non-small cell lung cancer in in vitro A549 cells.

Materials and methods: The anticancer effects of resveratrol were analyzed on cell viability, migration and invasion, proliferation and apoptosis. Cell viability was determined by sulphorhodamine B assays. Cell proliferation and apoptosis were determined by flow cytometry and migration and invasion by transwell chamber analysis. Expression of STAT-3 was examined by real-time polymerase chain reaction and western blot. Overexpressing vector of STAT-3 was also constructed and transfected into A549 cells to observe the effects of resveratrol on STAT-3 signaling.

Results: The results showed that resveratrol displayed a dose-dependent and time-dependent cytotoxicity action on A549 cell viability. Resveratrol also inhibited proliferation, migration and invasion and promoted apoptosis in a time-dependent manner from 0-72 hours. Further study showed that resveratrol inhibited the messenger RNA and protein expression of STAT-3, and overexpressed STAT-3 abolished the effects of resveratrol on proliferation, apoptosis, migration and invasion totally or in part.

Conclusions: These results suggest that the anticancer effects of resveratrol are mediated by STAT-3 signaling.

Keywords: A549 cells; Apoptosis; Proliferation; Resveratrol; STAT-3.

MeSH terms

  • A549 Cells
  • Antineoplastic Agents, Phytogenic / pharmacology
  • Antineoplastic Agents, Phytogenic / therapeutic use*
  • Apoptosis / drug effects
  • Carcinoma, Non-Small-Cell Lung / drug therapy*
  • Cell Movement / drug effects
  • Cell Proliferation / drug effects
  • Drug Screening Assays, Antitumor
  • Gene Transfer Techniques
  • Humans
  • Lung Neoplasms / drug therapy*
  • Resveratrol
  • STAT3 Transcription Factor / antagonists & inhibitors*
  • STAT3 Transcription Factor / genetics
  • STAT3 Transcription Factor / metabolism
  • Stilbenes / pharmacology
  • Stilbenes / therapeutic use*

Substances

  • Antineoplastic Agents, Phytogenic
  • STAT3 Transcription Factor
  • STAT3 protein, human
  • Stilbenes
  • Resveratrol