Abstract
Three antioxidant isoflavonoids characterized as 4',7,8-trihydroxyisoflavone (1), 3',4',7-trihydroxyisoflavone (2) and 8-chloro-3',4',5,7-tetrahydroxyisoflavone (3) were isolated from the cultured broth of Streptomyces sp. OH-1049. Among them, 3 is a novel isoflavonoid possessing a chlorine atom in the molecule. In in vitro studies, these antibiotics were found to possess antioxidant activity whereas showed almost no cytocidal activities against HeLa S3 cells.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Animals
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Anti-Bacterial Agents / isolation & purification*
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Anti-Bacterial Agents / pharmacology
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Antioxidants / isolation & purification*
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Antioxidants / pharmacology
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Fermentation
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Flavonoids / isolation & purification*
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HeLa Cells / drug effects
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Isoflavones / isolation & purification*
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Isoflavones / pharmacology
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Male
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Microbial Sensitivity Tests
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Rats
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Rats, Inbred Strains
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Streptomyces / classification
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Structure-Activity Relationship
Substances
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Anti-Bacterial Agents
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Antioxidants
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Flavonoids
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Isoflavones
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8-chloro-3',4',5,7-tetrahydroxyisoflavone
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4',7,8-trihydroxyisoflavone
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3',4',7-trihydroxyisoflavone