The in vitro biosynthesis of epitestosterone and testosterone from C19 steroid precursors in the testis of the lizard Tiliqua rugosa

Gen Comp Endocrinol. 1989 Aug;75(2):280-6. doi: 10.1016/0016-6480(89)90081-6.

Abstract

The metabolism of androgens in the testis of the lizard Tiliqua rugosa has been studied in vitro by incubating cellular homogenates with radiolabeled C19-steroid substrates. The identification 17 beta-oxidoreductase and 3 beta-hydroxysteroid dehydrogenase/isomerase activities. Aromatase, 5 alpha-reductase, and 17 alpha/beta-epimerase activities were not detected. The 17 alpha-oxidoreductase activity was temperature dependent (maximal at 32 degrees), while the 17 beta-oxidoreductase activity was temperature independent. Time yield and dual-label studies indicated that testosterone biosynthesis mainly involves the 4-ene pathway (via androstenedione), whereas the formation of epitestosterone uses both the 4-ene and 5-ene (via 5-androstene-3 beta, 17 alpha-diol) pathways. The function of alternative pathways in androgen biosynthesis is discussed, as is the role of temperature in the intratesticular regulation of androgen production.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Androstenediol / isolation & purification
  • Androstenediol / metabolism*
  • Androstenediols / metabolism*
  • Animals
  • Carbon Radioisotopes
  • Epitestosterone / biosynthesis*
  • Lizards
  • Male
  • Temperature
  • Testis / metabolism*
  • Testosterone / biosynthesis*
  • Tritium

Substances

  • Androstenediols
  • Carbon Radioisotopes
  • Tritium
  • Testosterone
  • Epitestosterone
  • Androstenediol