A Specific Gut Microbiota Dysbiosis of Type 2 Diabetic Mice Induces GLP-1 Resistance through an Enteric NO-Dependent and Gut-Brain Axis Mechanism

Cell Metab. 2017 May 2;25(5):1075-1090.e5. doi: 10.1016/j.cmet.2017.04.013.

Abstract

Glucagon-like peptide-1 (GLP-1)-based therapies control glycemia in type 2 diabetic (T2D) patients. However, in some patients the treatment must be discontinued, defining a state of GLP-1 resistance. In animal models we identified a specific set of ileum bacteria impairing the GLP-1-activated gut-brain axis for the control of insulin secretion and gastric emptying. Using prediction algorithms, we identified bacterial pathways related to amino acid metabolism and transport system modules associated to GLP-1 resistance. The conventionalization of germ-free mice demonstrated their role in enteric neuron biology and the gut-brain-periphery axis. Altogether, insulin secretion and gastric emptying require functional GLP-1 receptor and neuronal nitric oxide synthase in the enteric nervous system within a eubiotic gut microbiota environment. Our data open a novel route to improve GLP-1-based therapies.

Keywords: autonomic nervous system; enteric neurons; gut brain axis; incretins; metabolic diseases; microbiota; nitric oxide.

MeSH terms

  • Animals
  • Brain / metabolism*
  • Brain / pathology
  • Diabetes Mellitus, Type 2 / metabolism*
  • Diabetes Mellitus, Type 2 / microbiology
  • Diabetes Mellitus, Type 2 / pathology
  • Dysbiosis / metabolism*
  • Dysbiosis / microbiology
  • Dysbiosis / pathology
  • Enteric Nervous System / metabolism*
  • Enteric Nervous System / microbiology
  • Enteric Nervous System / pathology
  • Gastrointestinal Microbiome*
  • Gastrointestinal Tract / metabolism
  • Gastrointestinal Tract / microbiology
  • Gastrointestinal Tract / pathology
  • Glucagon-Like Peptide 1 / metabolism
  • Glucagon-Like Peptide-1 Receptor / metabolism
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Nitric Oxide / metabolism*

Substances

  • Glucagon-Like Peptide-1 Receptor
  • Nitric Oxide
  • Glucagon-Like Peptide 1