Thymidine phosphorylase promotes metastasis and serves as a marker of poor prognosis in hepatocellular carcinoma

Lab Invest. 2017 Aug;97(8):903-912. doi: 10.1038/labinvest.2017.51. Epub 2017 May 22.

Abstract

Hepatocellular carcinoma (HCC) ranks as one of the most common and lethal malignancies worldwide. A better understanding of the mechanism responsible for HCC metastasis will be helpful for the treatment of HCC patients. Thymidine phosphorylase (TP), a key enzyme that catalyzes the conversion of thymidine to thymine and deoxyribose-1-phosphate, was demonstrated to promote the invasion and metastasis of HCC in our study. Clinical retrospective analysis revealed that metastatic HCC tumor tissues have higher TP expression, and TP expression was significantly correlated with matrix metalloproteinase (MMP) 2 and 9 expression. Survival analysis revealed that TP expression was negatively correlated with the prognosis of HCC patients. Moreover, in vitro cell experiments confirmed that TP could promote the migration and invasion of HCC cells. In addition, MMP2 and MMP9 were activated by TP overexpression. Overall, this study suggests that TP promotes metastasis and may serve as a marker of poor prognosis in HCC. Thus, TP is a potential target for the treatment of HCC.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biomarkers, Tumor / analysis*
  • Carcinoma, Hepatocellular / diagnosis
  • Carcinoma, Hepatocellular / metabolism*
  • Carcinoma, Hepatocellular / mortality
  • Cell Movement / drug effects
  • Female
  • Humans
  • Immunohistochemistry
  • Liver Neoplasms / diagnosis
  • Liver Neoplasms / metabolism*
  • Liver Neoplasms / mortality
  • Male
  • Matrix Metalloproteinase 2 / metabolism
  • Matrix Metalloproteinase 9 / metabolism
  • Mice
  • Mice, Inbred BALB C
  • Middle Aged
  • Neoplasm Invasiveness / physiopathology
  • Prognosis
  • Retrospective Studies
  • Thymidine Phosphorylase / analysis
  • Thymidine Phosphorylase / metabolism*
  • Thymidine Phosphorylase / pharmacology
  • Xenograft Model Antitumor Assays

Substances

  • Biomarkers, Tumor
  • Thymidine Phosphorylase
  • Matrix Metalloproteinase 2
  • Matrix Metalloproteinase 9