Antihypertensive and renal effects of tertatolol, a new beta-blocking agent, in hypertensive patients

Am J Nephrol. 1986:6 Suppl 2:45-9. doi: 10.1159/000167333.

Abstract

Tertatolol, a new nonselective beta-adrenoceptor blocker, was administered to 11 hypertensive patients in a short-term study. Systolic and diastolic blood pressure and heart rate were significantly decreased when compared to the placebo period: in spite of that glomerular filtration rate and renal plasma flow were unchanged. The administration of metoclopramide (a dopaminergic receptor antagonist) caused a significant reduction of renal plasma flow and a significant rise of renal vascular resistances during placebo, but no change during tertatolol therapy. A possible interference of tertatolol on dopaminergic receptors is discussed as the mechanism responsible for the unmodified renal plasma flow despite the significant blood pressure lowering with tertatolol.

MeSH terms

  • Adrenergic beta-Antagonists / pharmacology*
  • Adult
  • Antihypertensive Agents / pharmacology*
  • Blood Pressure / drug effects
  • Female
  • Glomerular Filtration Rate / drug effects
  • Heart Rate / drug effects
  • Humans
  • Hypertension / physiopathology*
  • Kidney / drug effects*
  • Male
  • Metoclopramide / pharmacology
  • Middle Aged
  • Propanolamines / pharmacology*
  • Renal Circulation / drug effects
  • Renin / blood
  • Thiophenes*

Substances

  • Adrenergic beta-Antagonists
  • Antihypertensive Agents
  • Propanolamines
  • Thiophenes
  • tertatolol
  • Renin
  • Metoclopramide