Collapsing the Tumor Ecosystem: Preventing Adaptive Response to Treatment by Inhibiting Transcription

Cancer Discov. 2018 Jan;8(1):17-19. doi: 10.1158/2159-8290.CD-17-1245.

Abstract

<b/> Adaptation and resistance to treatment are the results of a multitude of (epi)genetic events unmasked or directly triggered by therapies targeting the genetic driver(s) of a dominant cell population within a tumor mass. Rusan and colleagues report that drug-tolerant cells are sensitive to THZ1, a dual CDK7/12 inhibitor, which, by impairing the transcriptional machinery, can prevent cellular rewiring to survive therapeutic attack. Cancer Discov; 8(1); 17-9. ©2018 AACRSee related article by Rusan et al., p. 59.

Publication types

  • Comment

MeSH terms

  • Ecosystem*
  • Humans
  • Neoplasms*