Pharmacotherapy for obesity in individuals with type 2 diabetes

Expert Opin Pharmacother. 2018 Feb;19(3):223-231. doi: 10.1080/14656566.2018.1428558. Epub 2018 Jan 29.

Abstract

Introduction: Type 2 diabetes (T2DM) is associated with significant morbidity and mortality. Obesity is one of the main risk factors for T2DM and its management requires a multidisciplinary approach, which may include pharmacotherapy.

Areas covered: In this paper, data on efficacy, tolerability and safety of FDA-approved pharmacotherapies for obesity (orlistat, phentermine/topiramate extended-release, lorcaserin, bupropion sustained release/naltrexone sustained release and liraglutide) are reviewed, focusing on individuals with type 2 diabetes.

Expert opinion: Obesity is the major pathophysiologic driver of T2DM; conversely 5-10% weight loss leads to significant improvement in glycemic control, lipids and blood pressure. Weight loss maintenance is difficult with lifestyle interventions alone and may require adjunctive therapies. There is good evidence for the efficacy and tolerability of approved anti-obesity pharmacotherapies in individuals with T2DM, with current cardiovascular safety data being most favorable for liraglutide, orlistat and lorcaserin. Given the link between obesity and T2DM, a weight-centric therapeutic approach including use of weight reducing anti-diabetic therapies, and anti-obesity pharmacotherapies is both intuitive and rational to improve glycemic and other metabolic outcomes in patients with T2DM.

Keywords: Obesity; pharmacotherapy; type 2 diabetes; weight loss.

Publication types

  • Review

MeSH terms

  • Anti-Obesity Agents / chemistry
  • Anti-Obesity Agents / pharmacology
  • Anti-Obesity Agents / therapeutic use*
  • Benzazepines / chemistry
  • Benzazepines / pharmacology
  • Benzazepines / therapeutic use
  • Clinical Trials as Topic
  • Diabetes Mellitus, Type 2 / complications*
  • Drug Compounding
  • Humans
  • Lactones / chemistry
  • Lactones / pharmacology
  • Lactones / therapeutic use
  • Liraglutide / chemistry
  • Liraglutide / pharmacology
  • Liraglutide / therapeutic use
  • Obesity / drug therapy*
  • Orlistat
  • Phentermine / chemistry
  • Phentermine / pharmacology
  • Phentermine / therapeutic use
  • Weight Loss / drug effects

Substances

  • Anti-Obesity Agents
  • Benzazepines
  • Lactones
  • lorcaserin
  • Liraglutide
  • Orlistat
  • Phentermine