Cancer vaccine formulation dictates synergy with CTLA-4 and PD-L1 checkpoint blockade therapy

J Clin Invest. 2018 Apr 2;128(4):1338-1354. doi: 10.1172/JCI93303. Epub 2018 Feb 26.

Abstract

Anticancer vaccination is a promising approach to increase the efficacy of cytotoxic T lymphocyte-associated protein 4 (CTLA-4) and programmed death ligand 1 (PD-L1) checkpoint blockade therapies. However, the landmark FDA registration trial for anti-CTLA-4 therapy (ipilimumab) revealed a complete lack of benefit of adding vaccination with gp100 peptide formulated in incomplete Freund's adjuvant (IFA). Here, using a mouse model of melanoma, we found that gp100 vaccination induced gp100-specific effector T cells (Teffs), which dominantly forced trafficking of anti-CTLA-4-induced, non-gp100-specific Teffs away from the tumor, reducing tumor control. The inflamed vaccination site subsequently also sequestered and destroyed anti-CTLA-4-induced Teffs with specificities for tumor antigens other than gp100, reducing the antitumor efficacy of anti-CTLA-4 therapy. Mechanistically, Teffs at the vaccination site recruited inflammatory monocytes, which in turn attracted additional Teffs in a vicious cycle mediated by IFN-γ, CXCR3, ICAM-1, and CCL2, dependent on IFA formulation. In contrast, nonpersistent vaccine formulations based on dendritic cells, viral vectors, or water-soluble peptides potently synergized with checkpoint blockade of both CTLA-4 and PD-L1 and induced complete tumor regression, including in settings of primary resistance to dual checkpoint blockade. We conclude that cancer vaccine formulation can dominantly determine synergy, or lack thereof, with CTLA-4 and PD-L1 checkpoint blockade therapy for cancer.

Keywords: Cancer immunotherapy; Immunology.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • B7-H1 Antigen / genetics
  • B7-H1 Antigen / immunology*
  • CTLA-4 Antigen / genetics
  • CTLA-4 Antigen / immunology*
  • Cancer Vaccines / immunology
  • Cancer Vaccines / pharmacology*
  • Cell Cycle Checkpoints / drug effects
  • Cell Cycle Checkpoints / genetics
  • Cell Cycle Checkpoints / immunology*
  • Cell Line, Tumor
  • Chemokine CCL2 / genetics
  • Chemokine CCL2 / immunology
  • Dendritic Cells / immunology
  • Dendritic Cells / pathology
  • Intercellular Adhesion Molecule-1 / genetics
  • Intercellular Adhesion Molecule-1 / immunology
  • Melanoma / genetics
  • Melanoma / immunology
  • Melanoma / pathology
  • Melanoma / therapy*
  • Mice
  • Mice, Transgenic
  • Monocytes / immunology
  • Monocytes / pathology
  • Neoplasms, Experimental / genetics
  • Neoplasms, Experimental / immunology
  • Neoplasms, Experimental / pathology
  • Neoplasms, Experimental / therapy*
  • Peptides / immunology*
  • Peptides / pharmacology
  • Receptors, CXCR3 / genetics
  • Receptors, CXCR3 / immunology
  • T-Lymphocytes, Regulatory / immunology
  • T-Lymphocytes, Regulatory / pathology
  • gp100 Melanoma Antigen / immunology
  • gp100 Melanoma Antigen / pharmacology*

Substances

  • B7-H1 Antigen
  • CTLA-4 Antigen
  • Cancer Vaccines
  • Ccl2 protein, mouse
  • Cd274 protein, mouse
  • Chemokine CCL2
  • Ctla4 protein, mouse
  • Cxcr3 protein, mouse
  • Icam1 protein, mouse
  • Peptides
  • Receptors, CXCR3
  • gp100 Melanoma Antigen
  • Intercellular Adhesion Molecule-1