Suspected drug-induced liver injury associated with iguratimod: a case report and review of the literature

BMC Gastroenterol. 2018 Aug 24;18(1):130. doi: 10.1186/s12876-018-0858-z.

Abstract

Background: Iguratimod is a novel anti-rheumatic drug with the capability of anti-cytokines as report goes. It has been reported that iguratimod is effective and safe for rheumatoid arthritis and other rheumatisms. As side effects, iguratimod can cause gastrointestinal reactions, dizziness, headache and itchy.

Case presentation: In this case report, a 60-year-old female patient was admitted with suspected drug-induced liver injury (DILI) caused by iguratimod. The causality assessment was done by the updated RUCAM, and the possibility of the case in our paper diagnosed as highly probable for the score was 9 points. Iguratimod was discontinued immediately, and methylprednisolone was used for acute liver injury and Sjogren's syndrome. The data showed the patient has improved gradually, and she was discharged on day 27. The true incidence of iguratimod-related hepatotoxicity and its pathogenic mechanism are largely unknown. It is difficult to recognize and diagnose DILI, and there is no standard for diagnosis of DILI. At the same time, the DILI is still lack of specific treatment.

Conclusions: Based on this rare case of severe liver injury, we recommend careful monitoring of liver function throughout iguratimod treatment for diseases.

Keywords: Clinical features; Drug-induced liver injury; Iguratimod; Pathogenesis; Treatment.

Publication types

  • Case Reports
  • Review

MeSH terms

  • Chemical and Drug Induced Liver Injury / drug therapy
  • Chemical and Drug Induced Liver Injury / etiology*
  • Chromones / adverse effects*
  • Female
  • Glucocorticoids / therapeutic use
  • Humans
  • Immunosuppressive Agents / adverse effects*
  • Methylprednisolone / therapeutic use
  • Middle Aged
  • Sjogren's Syndrome / drug therapy*
  • Sulfonamides / adverse effects*

Substances

  • Chromones
  • Glucocorticoids
  • Immunosuppressive Agents
  • Sulfonamides
  • iguratimod
  • Methylprednisolone