Sfrp5 increases glucose-stimulated insulin secretion in the rat pancreatic beta cell line INS-1E

PLoS One. 2019 Mar 28;14(3):e0213650. doi: 10.1371/journal.pone.0213650. eCollection 2019.

Abstract

Previous studies reported that secreted frizzled-related protein-5 (Sfrp5) decreases beta cell proliferation and increases fasting insulin levels, but studies on direct effects of Sfrp5 on insulin secretion and its underlying mechanisms are missing. This study examined effects of Sfrp5 on (i) beta cell viability and proliferation, (ii) basal and glucose-stimulated insulin secretion and (iii) canonical and non-canonical Wnt signalling pathways. We incubated rat INS-1E cells with 0.1, 1 or 5 μg/ml recombinant Sfrp5 for 24h. We measured basal and glucose-stimulated insulin secretion at glucose concentrations of 2.5 and 20 mmol/l. Phosphorylated and total protein content as well as mRNA levels of markers of cell proliferation, canonical and non-canonical Wnt signalling pathways were examined using Western blotting and real-time PCR. Differences between treatments were analysed by repeated measurement one-way ANOVA or Friedman's test followed by correction for multiple testing using the Benjamini-Hochberg procedure. At 5 μg/ml, Sfrp5 reduced mRNA levels of cyclin-B1 by 25% (p<0.05). At 1 and 5 μg/ml, Sfrp5 increased glucose-stimulated insulin secretion by 24% and by 34% (both p<0.05), respectively, but had no impact on basal insulin secretion. Sfrp5 reduced the phosphorylation of the splicing forms p46 and p54 of JNK by 39% (p<0.01) and 49% (p<0.05), respectively. In conclusion, Sfrp5 reduced markers of cell proliferation, but increased in parallel dose-dependently glucose-stimulated insulin secretion in INS-1E cells. This effect is likely mediated by reduced JNK activity, an important component of the non-canonical Wnt signalling pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adipokines / metabolism*
  • Animals
  • Blood Glucose / metabolism
  • Cell Line
  • Cell Proliferation
  • Cell Survival
  • Cyclin B1 / metabolism
  • Glucose / metabolism*
  • Insulin / metabolism*
  • Insulin Secretion*
  • Insulin-Secreting Cells / drug effects*
  • MAP Kinase Kinase 4 / metabolism
  • Phosphorylation
  • RNA, Messenger / metabolism
  • Rats
  • Signal Transduction
  • Wnt Proteins / metabolism
  • Wnt Signaling Pathway

Substances

  • Adipokines
  • Blood Glucose
  • Cyclin B1
  • Insulin
  • RNA, Messenger
  • Wnt Proteins
  • secreted frizzled-related protein 5, rat
  • MAP Kinase Kinase 4
  • Glucose

Grants and funding

This study was supported by research grants from the German Diabetes Association (Deutsche Diabetes-Gesellschaft, DDG) to MCK. This work was also supported by the Ministry of Culture and Science of the State of North Rhine-Westphalia and the German Federal Ministry of Health (BMG). This study was supported in part by a grant from the German Federal Ministry of Education and Research (BMBF) to the German Center for Diabetes Research (DZD). The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript.