Treatment of cancer with a combination of LAG-3Ig and anti-PD-1/anti-PD-L1 antibodies: a patent evaluation of US2018271940 A1

Expert Opin Ther Pat. 2019 May;29(5):311-314. doi: 10.1080/13543776.2019.1608947. Epub 2019 Apr 24.

Abstract

LAG-3 is checkpoint inhibitor in cancer that coordinates the down regulation of the proliferation of antigen-specific lymphocytes. There is a great need to discover and develop new therapies focused on inhibiting the action of LAG-3 and consequently improving the immune response in the various types of cancer. Authors of patent US2018271940 propose a method to eradicate cancer that utilizes the combination of LAG-3Ig and anti-PD-1 or anti-PD-L1 antibodies. Areas covered: Patent US2018271940 describes a method consisting of the utilization of either a pharmaceutical cocktail containing LAG-3Ig and an anti-PD-1 or anti-PD-L1 antibody for activation of T cells as a potential for the treatment of cancer. Expert opinion: Data supporting the patent demonstrate the ability of LAG-3Ig and PD-1/PD-L1 to be useful in T cells activation, in addition to the reports showing that LAG-3 and anti-PD-1 and PD-L1 antibodies are therapeutic agents against cancer. Although the proposed methodology is very interesting and promising, further studies are necessary to assess the clinical applicability of the inventions on cancer.

Keywords: LAG-3; cancer; checkpoint; immuno-oncology; immunotherapy; patent.

MeSH terms

  • Animals
  • Antibodies / administration & dosage*
  • Antibodies / immunology
  • Antigens, CD / immunology
  • B7-H1 Antigen / immunology
  • Humans
  • Immunotherapy / methods*
  • Lymphocyte Activation Gene 3 Protein
  • Neoplasms / immunology
  • Neoplasms / therapy*
  • Patents as Topic
  • Programmed Cell Death 1 Receptor / immunology
  • T-Lymphocytes / immunology

Substances

  • Antibodies
  • Antigens, CD
  • B7-H1 Antigen
  • CD274 protein, human
  • PDCD1 protein, human
  • Programmed Cell Death 1 Receptor
  • Lymphocyte Activation Gene 3 Protein
  • Lag3 protein, human
  • soluble LAG-3 protein, human